| View by Year: 2021, 2020, 2019,2018, 2017, 2016,2015, 2014,2013, 2012 2011, 2010, 2009, 2008, 2007, 2006, 2005, 2004, 2003, 2002,before 2002 |
| 2021 | Top | Concise Unified Access to (−)-8-Deoxy-13-dehydroserratinine,(+)-Fawcettimine, (+)-Fawcettidine, and (−)-8-DeoxyserratinineUsing a Direct Intramolecular Reductive Coupling Lin-Rui Zhong, Bing-Bing Huang, Xiao-Liang Yang, Shaozhong Wang, and Zhu-Jun Yao
Org. Lett. 2021, 23, 3578−3583.(DOI: 10.1021/acs.orglett.1c00977)

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| An Artemisinin Derivative ART1 Induces Ferroptosis by Targeting the HSD17B4 Protein Essential for Lipid Metabolism and Directly Inducing Lipid Peroxidation | Jingjing Xie, Guangya Zhu, Ming Gao, Jie Xi, Ge Chen, Xinxin Ma, Yu Yan, Zhiyuan Wang, Ze-Jun Xu, Hui-Jun Chen, Hong-Dong Hao, Yaoyang Zhang, Zhu-Jun Yao and Jidong Zhu | CCS Chem. 2021,3, 664–677.(DOI: org/10.31635/ccschem.021.202000691)
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| Diastereoselective Access to Tetracyclic Eight-Membered Lactams through a Dearomative Heck Reaction and an Alkylative RingOpening Driven by Photoexcited Spiroindoline | Jianhui Qiao, Wenxuan Zhao, Yong Liang, Zhu-Jun Yao, and Shaozhong Wang | Chem. Eur. J. 2021, 27, 6308 – 6314.(DOI: org/10.1002/chem.202005369) | 
A gram-scale laboratory synthesis of Annonaceous acetogenin mimic AA005
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| Baobao Yu, Zhu-Jun Yao Chinese Chemical Letters. 2021. 32. 408–412.

Scalable Cu(II)-mediated intramolecular dehydrogenative phenol-phenol coupling: Concise synthesis of enantiopure axially chiral homo- and hetero-dephenols
Yuefei Gu, Tianyang Wang, Ming Gao, Zhu-Jun Yao
Chinese Chemical Letters, 2021, 32(1): 380-384.(DOI:10.1016/j.cclet.2020.02.015)

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| 2020 | Top |
| YL064 activates proteasomal-dependent degradation of c-Myc and synergistically enhances the anti-tumor activity of ABT-199 in diffuse large B cell lymphoma | Huizhuang Shan, Yang Cao, Xinhua Xiao, Meng Liu, Yunzhao Wu, Qi Zhu, Hanzhang Xu, Hu Lei, Zhujun Yao, and Yingli Wu | Signal Transduction and Targeted Therapy . 2020, 5, 116; https://doi.org/10.1038/s41392-020-00236-1. |
| New triterpenoid saponin glycosides from the fruit fibers of Trichosanthes cucumerina L. | Parichat Suebsakwong, Wanatsanan Chulrik, Warangkana Chunglok, Jian-Xin Li, Zhu-Jun Yao, and Apichart Suksamrarn | RSC Adv. 2020, 10, 10461-10470.(DOI:10.1039/d0ra01176b) | 
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| An eight-step total synthesis of pyrroloquinolone-type Lycopodium alkaloid via a tandem annulation approach |
| Lin-Rui Zhong, Yuanjie Yang, Bing-Bing Huang, and Zhu-Jun Yao |
| Chin. J. Chem. 2020, 38, 10.1002/cjoc.202000273. |
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| 2019 | Top |
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| Diastereoselective Synthesis of Polysubstituted Piperidines via Visible Light-Driven Silylative Cyclization of Aza-1,6-Dienes: Experimental and DFT Studies |
| Wei-Chen Cui, Wenxuan Zhao, Ming Gao, Wei Liu, Shaozhong Wang, Yong Liang and Zhu-Jun Yao |
| Chem. Eur. J. 10.1002/chem.201903440.(DOI:10.1002/chem.201903440) |
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| A Bioreductive Prodrug of Cucurbitacin B Significantly Inhibits Tumor Growth in the 4T1 Xenograft Mice Model |
| Parichat Suebsakwong, Jie Wang, Phorntip Khetkam, Natthida Weerapreeyakul, Jing Wu, Yun Du, Zhu-Jun Yao, Jian-Xin Li, and Apichart Suksamrarn |
| ACS Med. Chem. Lett. 2019, 10, 1400-1406.(DOI:10.1021/acsmedchemlett.9b00161) |
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| Divergent Synthesis of Oxa-Cyclic Nitrones through Gold(I)-Catalyzed 1,3-Azaprotio Transfer of Propargylic α-Ketocarboxylatte Oximes:Experimental and DFT Studies |
| Chunhong Wang, Qi Cui, Zhixin Zhang, Zhu-Jun Yao, Shaozhong Wang, Zhi-Xiang Yu |
| Chem. Eur. J. 2019, 25, 9821-9826.(DOI:10.1002/chem.201901522). |
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| 2018 | Top |
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| Visible Light-Driven Radical trans-Hydrosilylation of Electron-Neutral and -Rich Alkenes with Tertiary and Secondary Hydrosilanes |
| Jing Zhu, Wei-Chen Cui, Shaozhong Wang, and Zhu-Jun Yao |
| J. Org. Chem. 2018, 83,14600-14609.(DOI:10.1021/acs.joc.8b02409) |
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| 11‐Aza‐artemisinin Derivatives Exhibit Anticancer Activities by Targeting the Fatty Acid Binding Protein 6 (FABP6) |
| Xin-Ya Chen, Yue Yin, Jie Xi, Yi Yuan, Yan Li, Qing Li, Ren-Xiao Wang, Zhu-Jun Yao, Gong-Li Tang |
| Chin. J. Chem. 2018, 36, 1197-1201.(DOI:10.1002/cjoc.201800361) |
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| YL064 directly inhibits STAT3 activity to induce apoptosis of multiple myeloma cells |
| Yingying Wang, Linlin Wu, Haiyan Cai, Hu Lei, Chun-Min Ma, Li Yang, Hanzhang Xu, Qi Zhu, Zhujun Yao and Yingli Wu |
| Cell Death Discovery. 2019, 5, 44(DOI 10.1038/s41420-018-0108-8) |
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| Total Synthesis of (+)-Plumisclerin A |
| Ming Gao,Ye-Cheng Wang,Kai-Rui Yang,Wei He,Xiao-Liang Yang,and Z.-J Yao |
| Angew. Chem. Int. Ed. 2018, 57, 13313-13318. (DOI:10.1002/anie.201808517) |
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| Annonaceous acetogenin mimic AA005 suppresses human colon cancer cell growth in vivo through downregulation of Mcl-1 |
| Bing Han, Yu-xia Cao, Zhan-ming Li, Zhao-xia Wu, Yu-qin Mao, Hui-ling Chen, Zhu-jun Yao and Li-shun Wang |
| Acta Pharmacologica Sinica. 2018, 0, 1–12(DOI:10.1038/s41401-018-0025-7) |
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| Efficiency in Natural Product Total Synthesis |
| Pei-Qiang Huang, Zhu-Jun Yao, Richard P.Hsung |
| ISBN-13:9781118940211(DOI:10.1002/9781118940228) |
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| Radical Hydrosilylation of Alkynes Catalyzed by Eosin Y and Thiol under Visible Light Irradiation |
| Jing Zhu,Wei-Chen Cui,Shaozhong Wang,and Zhu-Jun Yao |
| Org. Lett.2018, 20, 3174−3178 (DOI: 10.1021/acs.orglett.8b00909) |
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| 2017 | Top |
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| Synthesis of 2,3-Dialkylated Tartaric Acid Esters via Visible Light Photoredox-Catalyzed Reductive Dimerization of α-Ketoesters |
| Jing Zhu, Yi Yuan, Shaozhong Wang, and Zhu-Jun Yao |
| ACS Omega. 2017, 2, 4665−4677(DOI:10.1021/acsomega.7b00749) |
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| Recent advances in direct dehydrogenative biphenyl couplings |
| |
| SCIENCE CHINA Chemistry.2017. 60, 701-720(DOI:10.1007/s11426-016-0435-5) |
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| Azepinoindole Synthesis via a N‑Bromosuccinimide-Induced Cycloisomerization of Enaminoester/Enaminone |
| Lina Chang, Tao Guo, Ziyi Wang, Shaozhong Wang,and Zhu-Jun Yao |
| J. Org. Chem.2017, 82, 1567−1574 (DOI: 10.1021/acs.joc.6b02760) |
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| Nodupetide, a potent insecticide and antimicrobial from Nodulisporium sp. associated with Riptortus pedestris |
| Hui Min Wu, Li Ping Lin, Qin Lan Xu, Wen Bo Han, Song Zhang, Ze Wen Liu, Ya Ning Mei,Zhu Jun Yao,and Ren Xiang Tan |
| Tetrahedron Letters. 2017, 58, 663–665(DOI.org/10.1016/j.tetlet.2017.01.009) |
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| 2016 | Top |
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| Michael addition-based cyclization strategy in the total synthesis of Lycopodium alkaloids |
| Lin-Rui Zhong and Yao Zhu-Jun* |
| SCIENCE CHINA Chemistry. 2016. 59. 1079-1087(DOI:10.1007/s11426-016-0056-0) |
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| Gram-Scale Laboratory Synthesis of UM171, a Potent Agonist of Human Hematopoietic Stem Cell Self-Renewal |
| Sajjad Ali, Shun-Ming Yu, and Zhu-Jun Yao* |
| J. Org. Chem.2016, 81, 10236−10241(DOI:10.1021/acs.joc.6b01094) |
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| Aerobic a-hydroxylation of b-keto esters and amides by co-catalysis of SmI3and I2 under mild base-free conditions |
| Shun-Ming Yu, Kai Cui, Fei Lv , Zhen-Yu Yang*, Zhu-Jun Yao* |
| Tetrahedron. Letters. 2016. 57. 2818-2821(DOI:10.1016/j.tetlet.2016.05.052) |
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| Convenient One-Step Synthesis of Benzo[c]phenanthridines by Three-Component Reactions of Isochromenylium Tetrafluoroborates and Stilbenes in Acetonitrile |
| Gang-Gang Chen, Jun-Qiang Wei, Xiaoliang Yang*, and Zhu-Jun Yao* |
| Org. Lett. 2016, 18, 1502–1505 (DOI: 10.1021/acs.orglett.6b00010) |
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| Enantioselective Total Synthesis of Lycoposerramine-Z Using Chiral Phosphoric Acid Catalyzed Intramolecular Michael Addition |
| Lan-De Zhang, Lin-Rui Zhong, Jie Xi, Xiao-Liang Yang*, and Zhu-Jun Yao* |
| J. Org. Chem. 2016, 81, 1899–1904 (DOI: 10.1021/acs.joc.5b02723) |
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| 2015 | Top |
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| Kinetic or Dynamic Control on a Bifurcating Potential Energy Surface?An Experimental and DFT Study of Gold-Catalyzed Ring Expansion and Spirocyclization of 2-Propargyl-β-tetrahydrocarbolines |
| Zhang Lei,Yi Wang,Yao Zhu-Jun,Wang Shao-Zhong,Yu Zhi-Xing |
| J. Am. Chem. Soc. 2015, 137, 13290–13300(DOI:10.1021/jacs.5b05971) |
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| Synthesis of Tricyclo[4,3,1,01,5]decane Core of Plumisclerin A Using Pauson–Khand Annulation and SmI2-Mediated Radical Cyclization |
| Chen Ji-Peng,He Wei,Yang Zhen-Yu,and Yao Zhu-Jun |
| Org. Lett. 2015, 17, 3379–3381(DOI:10.1021/acs.orglett.5b01563) |
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| Efficient Synthesis of Octahydrophenanthrene Derivatives with Mild Cascade Reactions of Isochromenylium Tetrafluoroborates and Bifunctional Styrenes , |
| Mo Lei, Wu Lin-Lin, Wang Shao-Zhong, Yao Zhu-Jun |
| Org. Lett. 2015, 17, 3314–3317(DOI:10.1021/acs.orglett.5b01532) |
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| The last and next decades of the Asian Core Program on cutting-edge organic chemistry in Asia |
| Minoru Isobe, Atsushi Nishida, Yeun-Mun Choo, Noorsaadah Abd. Rahman, Poonsakdi Ploypradith, Somsak Ruchirawat, Guo-Qiang Lin, Ang Li, Zhu-Jun Yao, Biing-Jiun Uang, Chun-Chen Liao, Pauline Chiu, Byeong Moon Kim, Teck Peng Loh |
| Chemistry - An Asian Journal.2015, 10, 790-804 |
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| Annonaceous acetogenin mimic AA005 induces cancer cell death via apoptosis inducing factor through a caspase-3-independent mechanism |
| Han Bing, Wang Tong-Dan, Shen Shao-Ming, Yu Yun, Mao Chan, Yao Zhu-Jun, Wang Li-Shun |
| BMC Cancer 2015, 15, 139 |
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| Short Protecting Group-free Syntheses of Camptothecin and 10-Hydroxycamptothecin Using Cascade Methodologies |
| Xu Peng, Chen Dong-Sheng Chen, Xi Jie, Yao Zhu-Jun |
| Chemistry - An Asian Journal.2015, 10, 976-981 |
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| Stereodivergent total synthesis of chlorofusin and its all seven chromophore diastereomers |
| Qiu Hai-Bo, Qian Wen-Jian, Yu Shun-Ming, Yao Zhu-Jun |
| Tetrahedron2015, 71, 370-380 |
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| 2014 | Top |
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| Total Synthesis of Ascididemin-Type Alkaloids Using Alkyne Building Blocks |
| Yin Hao, Shan Naiyu, Wang Shaozhong, Yao Zhu-Jun |
| Journal of Organic Chemistry .2014, 79, 9748-9753 |
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| Total synthesis of proposed structure of coibamide A, a highly N- and O-methylated cytotoxic marine cyclodepsipeptide |
| He Wei, Qiu Hai-Bo, Chen Yi-Jie, Xi Jie, Yao Zhu-Jun |
| Tetrahedron Letters.2014, 55, 6109-6112 |
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| Unified flexible total synthesis of chlorofusin and artificial Click mimics as antagonists against p53–HDM2 interactions |
| Qiu Hai-Bo, Chen Xin-Ya, Li Qing, Qian Wen-Jian, Yu Shun-Ming, Tang Gong-Li, Yao Zhu-Jun |
| Tetrahedron Letters.2014, 55, 6055-6059 |
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| Total Syntheses of Lycoposerramine-V and 5-epi-Lycoposerramine-V |
| Zhang Lan-De, Zhou Ting-Ting, Qi Sen-Xing, Xi Jie, Yang Xiao-Liang, Yao Zhu-Jun |
| Chemistry - An Asian Journal.2014, 9, 2740-2744 |
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| Asymmetric Annulation of 3‑Alkynylacrylaldehydes with Styrene-Type Olefins by Synergetic Relay Catalysis from AgOAc and Chiral Phosphoric Acid |
| Zhang Hao, Zhu Le, Wang Shaozhong, Yao Zhu-Jun |
| Journal of Organic Chemistry,2014, 79, 7063-7074 |
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| Regio-controlled synthesis of unsymmetrical pyrazine-fused sinomenine derivatives and discriminate substitution effects on TNF-α inhibitory activity |
| Zhou Tingting, Hou Jian, Wang Meng, Ma Liyan, Wu Linlin, Wang Shaozhong, Sun Bing, Yao Zhu-Jun |
| Tetrahedron2014.70. 5475-5482 |
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| New cytotoxic annonaceous acetogenin mimetics having a nitrogen-heterocyclic terminal and their application to cell imaging |
| Chen Yi-Jie, Jin Sheng, Xi Jie, Yao Zhu-Jun |
| Tetrahedron2014.70. 4921-4928 |
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| Total synthesis of ent-(−)-azonazine using a biomimetic direct oxidative cyclization and structural reassignment of natural product |
| Zhao Ji-Chen,Yu Shun-Ming,Qiu Hai-Bo,Yao Zhu-Jun |
| Tetrahedron.2014.70. 3197–3210 |
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| Biological evaluation of new mimetics of annonaceous acetogenins: Alteration of right scaffold by click linkage with aromatic functionalities |
| Liu Yanghan, Xiao Qicai, Liu Yongqiang, Li Zheng, Qiu Yatao, Zhou Guang-Biao, Yao Zhu-Jun, Jiang Sheng |
| European Journal of Medicinal Chemistry.2014. 78. 248-258 |
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| Identification of novel bivalent mimetics of annonaceousacetogenins via a scaffold-hopping strategy |
| Liu Yanghan, Liu Yongqiang, Li Zhen, Zhou Guang-Biao, Yao Zhu-Jun, Jiang Sheng |
| Bioorganic & Medicinal Chemistry Letters. 2014.24. 1650-1653 |
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| Azocinoindole Synthesis by a Gold(I)-Catalyzed Ring Expansion of2-Propargyl-b-Tetrahydrocarboline |
| Zhang Lei,ChangLina, Hu Hongwen, Wang Huaqin, Yao Zhu-Jun, Wang Shaozhong |
| Chemistry - A European Journal.2014,20, 2925-2932 |
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| 2013 | Top |
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| Assembly of indolo[1,2-c]quinazolines using ZnBr2-promoted domino hydroamination–cyclization |
| Xu Min, Xu Ke, Wang Shaozhong, Yao Zhu-Jun |
| Tetrahedron Letters,2013, 54, 4675-4678 |
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| 适用于荧光成像的化学发色团与生物正交反应研究进展 |
| 张艳, 陈鹏, 姚祝军 |
| Chinese Science Bulletin,2013, 58, 2872-2885 |
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| Synthesis of 2-vinyl-2H-benzotriazoles via NIS-promoted regio/stereoselective addition of 1H-benzotriazole to alkynes |
| Zhang ZhenHua, Chang Lina, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun |
| RSC Advances, 2013,3, 18446-18452 |
| 
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| Biomimetic Synthesis of ent-(−)-Azonazine and Stereochemical Reassignment of Natural Product |
| Zhao Ji-Chen, Yu Shun-Ming, Liu Yun, Yao Zhu-Jun |
| Organic Letters,2013, 15, 4300-4303 |
| 
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| Asymmetric Cascade Annulation Based on Enantioselective OxaDiels−Alder Cycloaddition of in Situ Generated Isochromenyliums by Cooperative Binary Catalysis of Pd(OAc)2 and (S)‑Trip |
| Yu Shu-Yan, Zhang Hao, Gao Yang, Mo Lei, Wang Shaozhong, Yao Zhu-Jun |
| Journal of the American Chemical Society, 2013, 135, 11402-11407 |
| 
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| Asymmetric Michael addition of 4H-thiopyran-4-one to nitroolefins catalyzed by diamine mono-N-sulfonamide and its application to concise synthesis of enantiopure multiring heterocycles |
| Mo Lei, Tang Huang, Yao Zhu-Jun |
| Tetrahedron, 2013, 69, 6897-6905 |
| 
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| Dual-Functional abeo-Taxane Derivatives Destabilizing Microtubule Equilibrium and Inhibiting NF-κB Activation |
| Yu Zhao, Jia Su, Masuo Goto, Susan L. Morris-Natschke, Yan Li, Qin-Shi Zhao, Zhu-Jun Yao, Kuo-Hsiung Lee |
| Journal of Medicinal Chemistry, 2013, 56, 4749−4757 |
| 
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| Asymmetric One-Pot Sequential Mannich/Hydroamination Reaction by Organo- and Gold Catalysts: Synthesis of Spiro[pyrrolidin-3,2′-oxindole] Derivatives |
| Chen Xianjie, Chen Hui, Ji Xun, Jiang Hualiang, Yao Zhu-Jun, Liu Hong |
| Organic Letters,2013, 15, 1846–1849 |
| 
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| Organocatalytic enantioselective conjugate addition of 2-nitrocyclohexanone to acrylaldehyde: a concise two-step synthesis of chiral building block 1-azaspiro[4.5]decan-6-one |
| Ding Xiao-Hua, Cui Wei-Chen, Li Xiang, Ju Xuan, Liu Dan, Wang Shaozhong, Yao Zhu-Jun |
| Tetrahedron Letters,2013, 54, 1956-1959 |
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| Assembly of fused indenes via Au(I)-catalyzed C1–C5 cyclization of enediynes bearing an internal nucleophile |
| Hou Qiwen, Zhang Zhenhua, Kong Fanji, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun |
| Chemical Communications,2013, 49, 695-697. |
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| 2012 | Top |
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| Sinomenine derivatives with embedment of nitrogen-containing heterocycles exhibiting potent TNF-αinhibitory activity |
| Wang Meng, Ma Li-Yan, Lou Yang-Tong, Bian Chao, Zhou Ting-Ting, Zhou Hai-Bin, Liao Hong-Ze, Ma Zhao, Yin Dong-Sheng, Wang Shaozhong, Yang Zhen-Yu, Sun Bing, Yao Zhu-Jun |
| Science China Chemistry,2012, 55, 2537-2547. |
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| Assembly of pentacyclic pyrido[4,3,2-mn]acridin-8-ones via a domino reaction initiated by Au(I)-catalyzed 6-endo-dig cycloisomerization of N-propargylaminoquinones |
| Yin Hao, Kong Fanji, Wang Shaozhong, Yao Zhu-Jun |
| Tetrahedron Letters,2012, 53, 7078-7082. |
| 
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| Gefitinib Analogue V1801 Induces Apoptosis of T790M EGFR-Harboring Lung Cancer Cells by Up-Regulation of the BH-3 Only Protein Noxa |
| Zhang Bo, Jiao Jiao, Liu Ying, Guo Liang-Xia, Zhou Bo, Li Gang-Qin, Yao Zhu-Jun, Zhou Guang-Biao |
| PLOS ONE,2012, 7(11), e48748. |
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| Identification of an Annonaceous Acetogenin Mimetic, AA005, as an AMPK Activator and Autophagy Inducer in Colon Cancer Cells |
| Liu Yong-Qiang, Cheng Xin, Guo Liang-Xia, Mao Chan, Chen Yi-Jie, Liu Hai-Xia, Xiao Qi-Cai, Jiang Sheng, Yao Zhu-Jun, Zhou Guang-Biao |
| PLOS ONE,2012, 7(10), e47049. |
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| Highly Enantioselective Michael Addition of 2-Oxindole- 3-carboxylate Esters to Nitroolefins Promoted by Cinchona Alkaloid-Thiourea-Brønsted Acid Cocatalysts |
| Chen Xian-Jie, Zhu Wei, Qian Wangke, Feng Enguang, Zhou Yu, Wang Jinfang, Jiang Hualiang, Yao Zhu-Jun, Liu Hong |
| Advanced Synthesis & Catalysis,2012, 354, 2151-2156. |
| 
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| Protecting Group-Free Total Synthesis of (−)-Lannotinidine B |
| Ge Hui-Ming, Zhang Lan-De, Tan Ren-Xiang, Yao Zhu-Jun |
| Journal of the American Chemical Society,2012, 134, 12323-12325. |
| 
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| Effect of Annonaceous Acetogenin Mimic AA005 on Proliferative Inhibition of Leukemia Cells in vitro and Its Possible Mechanisms |
| Han Bing, Yao Zhu-Jun, Wang Li-Shun |
| Journal of Experimental Hematology,2012, 20, 549-553. |
| 
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| Enantioselective Total Synthesis of Marine Diterpenoid Clavulactone |
| Yang Zhen-Yu, Liao Hong-Ze, Shen Kang, Chen Yong-Fei, Yao Zhu-Jun |
| Angewandte Chemie International Edition,2012, 51, 6484-6487. |
| 
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| Target-oriented multifunctional organocatalysis for enantioselective synthesis of bicyclo[3.3.1]nona-2,6-dien-9-ones. A formal asymmetric synthesis of huperzine A |
| Ding Xiao-Hua, Li Xiang, Liu Dan, Cui Wei-Chen, Ju Xuan, Wang Shaozhong, Yao Zhu-Jun |
| Tetrahedron,2012, 68, 6240-6248. |
| 
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| A simple selective protocol for continuous two-stage fluorescent sensing of both MeHg+ and anti-MeHg+ agents in living cells |
| Mei De-Sheng, He Bao-Kun, Chen Lei, Yao Zhu-Jun |
| Tetrahedron Letters,2012, 53, 3463-3466. |
| 
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| Brönsted acid-promoted dimerization of o-alkynylbenzaldehydes: a one-step synthesis of functionalized Kagan’s ether analogues |
| Zhang Hao, Cui Wei-Chen, Hu Zhi-Long, Yu Shu-Yan, Wang Shaozhong, Yao Zhu-Jun |
| RSC Advances,2012, 2, 5101-5104. |
| 
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| Electronically unfavorable addition of electron-deficient olefins to isochromenylium tetrafluoroborates initiated by C-1 O-glycosylation |
| Yu Shu-Yan, Hu Zhi-Long, Zhang Hao, Wang Shaozhong, Yao Zhu-Jun |
| Tetrahedron Letters,2012, 53, 2765-2768. |
| 
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| Regio- and stereoselective C10β–H functionalization of sinomenine: an access to more potent immunomodulating derivatives |
| Lou Yang-Tong, Ma Li-Yan, Wang Meng, Yin Dongsheng, Zhou Ting-Ting, Chen Ai-Zhong, Ma Zhao, Bian Chao, Wang Shaozhong, Yang Zhen-Yu, Sun Bing, Yao Zhu-Jun |
| Tetrahedron,2012, 68, 2172-2178. |
| 
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| Concise synthesis of zanamivir and its C4-thiocarbamido derivatives utilizing a [3+2]-cycloadduct derived from d-glucono-δ-lactone |
| Zhu Xue-Bin, Wang Meng, Wang Shaozhong, Yao Zhu-Jun |
| Tetrahedron,2012, 68, 2041-2044. |
| 
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| 2011 | Top |
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| Development of Novel Conformation-Constrained Cytotoxic Derivatives of Cheliensisin A by Embedment of Small Heterocycles |
| Deng Xu, Su Jia, Zhao Yu, Peng Li-Yan, Yao Zhu-Jun, Zhao Qin-Shi |
| European Journal of Medicinal Chemistry,2011, 46, 4238-4244. |
| 
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| Total Synthesis of 7-Ethyl-10-hydroxycamptothecin (SN38) and its Application to the Development of C18-Functionalized Camptothecin Derivativesivatives |
| Yao Yuan-Shan, Liu Jia-Li, Xi Jie, Miu Bukeyan, Liu Guan-Sai, Wang Shaozhong, Meng Linghua, Yao Zhu-Jun |
| Chemistry- A European Journal,2011, 17, 10462-10469. |
| 
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| Modular assembly of cytotoxic acetogenin mimetics by click linkage with nitrogen functionalities |
| Mao Chan, Han Bing, Wang Li-Shan, Wang Shaozhong, Yao Zhu-Jun |
| MedChemComm,2011, 2, 918-922. |
| 
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| CuCl(2)-Promoted 6-endo-dig Chlorocyclization and Oxidative Aromatization Cascade: Efficient Construction of 1-Azaanthraquinones from N-Propargylaminoquinones |
| Fei Na, Yin Hao, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun |
| Organic Letters,2011, 13, 4208-4211. |
| 
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| Efficient synthesis of furoquinolinones using Hendrickson reagent-initiated cascade annulation |
| Xu Peng, Liu Guan-Sai, Xi Jie, Wang Shaozhong, Yao Zhu-Jun |
| Tetrahedron,2011, 67, 5455-5460. |
| 
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| Generation of trans-arachidonic acid under nitrative stress is associated with upregulation of thromponsdin-1 in diabetic rats |
| Xu Lin, Liu Yu-Min, Yao Zhu-Jun, Xun Guo-Liang, Yu Wen-Juan, Liu Kun, Sun Xiao-Dong, Qiu Yun-Ping, Wu Hai-Xiang, Xu Xun |
| Chinese Medical Journal,2011, 124, 1885-1889. |
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| Evaluation of nitrative stress on retinal capillary by detection of trans-arachidonic acid with GC/MS in diabetic rats |
| Xu Lin, Xun Guo-Liang, Yao Zhu-Jun, Liu Yu-Min, Fan Ying, Sun Tao, Xu Xun |
| Chinese Journal of Experimental Ophthalmology,2011, 29, 432-436. |
|
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| Design, synthesis of symmetrical bivalent analogues mimetics of annonaceous acetogenins and their cytotoxicities |
| Xiao Qi-Cai, Liu Yong-Qiang, Qiu Ya-Tao, Yao Zhi-Yi, Zhou Guang-Biao, Yao Zhu-Jun, Jiang Sheng |
| Bioorganic & Medicinal Chemistry Letters,2011, 21, 3613-3615. |
| 
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|
| Study on Iron-Catalyzed Oxidative Free Radical Dimerization of Isochromenylium Tetrafluoroborate |
| Song Xiao-Nan, Mo Lei, Hu Zhi-Long, Yang Zhen-Yu, Yao Zhu-Jun |
| Acta Chimica Sinica,2011, 69, 680-686. |
|
|
| Syntheses and characterizations of novel pyrrolocoumarin probes for SNAP-tag labeling technology |
| Mei De-Sheng, Qu Yi, He Jin-Xiang, Chen Lei, Yao Zhu-Jun |
| Tetrahedron,2011, 67, 2251-2259. |
| 
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| Facile Assembly of 11H-Indolo[3,2-c]quinoline by a Two-Step Protocol Involving a Regioselective 6-endo-Cyclization Promoted by the Hendrickson Reagent |
| Xu Min, Hou Qiwen, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun |
| Synthesis-Stuttgart,2011, 4, 626-634. |
|
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| Potent Antitumor Mimetics of Annonaceous Acetogenins Embedded with an Aromatic Moiety in the Left Hydrocarbon Chain Part |
| Xiao Qi-Cai, Liu Yong-Qiang, Qiu Ya-Tao, Zhou Guang-Biao, Mao Chan, Li Zheng, Yao Zhu-Jun, Jiang Sheng |
| Journal of Medicinal Chemistry,2011, 54, 525-533. |
| 
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| Fragmentations of 13-oxo-taxyunnansin A and their application to preparation of abeo-paclitaxel and abeo-docetaxel analogues |
| Zhao Yu, Zhang Hong-Bin, Liu Ji-Kai, Su Jia, Li Yan, Yao Zhu-Jun, Zhao Qin-Shi |
| Tetrahedron Letters,2011, 52, 139-142. |
| 
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| Three-Component Reactions of Isochromenylium Tetrafluoroborates via Non-Classical [4+2]-Intermediates: Mild One-Step Metal-Free Synthesis of Functionalized Dihydronaphthalenes and Tetrahydronaphthalenes |
| Hu Zhi-Long, Yang Zhen-Yu, Wang Shaozhong, Yao Zhu-Jun |
| Chemistry-A European Journal,2011, 17, 1268-1274. |
| 
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| 2010 | Top |
|
|
| Synthesis of Tetrahydroisoquinolines via Cascade Reductive Amination of Isochromenylium Tetrafluoroborate with Primary Amines |
| Liao Hong-Ze, Hu Zhi-Long, Cui Kai, Jiao Jiao, Qin Yong, Yao Zhu-Jun |
| Synthesis-Stuttgart,2010, 20, 3474-3480. |
|
|
| Efficient Synthesis of Phenanthridines Using Hendrickson Reagent Initiated Cascade Reaction under Mild Conditions |
| Xi Jie, Dong Qing-Li, Liu Guan-Sai, Wang Shaozhong, Chen Lin, Yao Zhu-Jun |
| Synlett,2010, 11, 1674-1678. |
|
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| Efficient Synthesis of Phenanthridines Using Hendrickson Reagent Initiated Cascade Reaction under Mild Conditions |
| Jiang Chun-Hui, Xu Min, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun |
| Journal of Organic Chemistry,2010, 75, 4323-4325. |
| 
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| Synthesis of the cyclic nonapeptide of chlorofusin using a convergent [3+3+3]-fragment coupling strategy |
| Wang Yan-Li, Qian Wen-Jian, Wei Wan-Guo, Zhang Yue, Yao Zhu-Jun |
| Tetrahedron,2010, 66, 3427-3432. |
| 
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| Short asymmetric synthesis of (S,S)-PDP using L-prolinol derivative as economic starting material |
| Song Xiao-Nan, Yao Zhu-Jun |
| Tetrahedron,2010, 66, 2589-2593. |
| 
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|
| Direct nucleophilic C-1 addition of stable isochromenylium tetrafluoroborates under catalyst-free conditions: A new access to 1H-isochromenes |
| Hu Zhi-Long, Qian Wen-Jian, Yao Zhu-Jun |
| Science China-Chemistry,2010, 53, 869-876. |
|
|
| Total Synthesis of Chloptosin, a Potent Apoptosis-Inducing Cyclopeptide |
| Yu Shun-Ming, Hong Wen-Xu, Wu Yuan, Zhong Chun-Long, Yao Zhu-Jun |
| Organic Letters,2010, 12, 1124-1127. |
| 
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|
| Modification of poorly bioactive sinomenine into more potent immunosuppressive agents by embedding of drug-like fragments |
| Lou Yang-Tong, Zhou Hai-Bin, Zou Jia, Yan Ling-Chen, Bi En-Guan, Sun Bing, Yao Zhu-Jun |
| Tetrahedron Letters,2010, 51, 485-488. |
| 
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| Azaanthraquinone assembly from N-propargylamino quinone via iodine-induced 6-endo-dig electrophilic cyclization |
| Fei Na, Hou Qi-Wen, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun |
| Organic & Biomolecular Chemistry,2010, 8, 4096-4103. |
| 
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|
| Efficient Total Synthesis of (S)-14-Azacamptothecin |
| Liu Guan-Sai, Yao Yuan-Shan, Xu Peng, Wang Shaozhong, Yao Zhu-Jun |
| Chemistry-An Asian Journal,2010, 5, 1382-1388. |
| 
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| Synthesis of N(11)-anchoring biotinylated artemisinin derivatives and their preliminary biological assessment |
| Pan Qi-Yu, Wang Shaozhong, Lu JinJian, Meng Linghua, Yao Zhu-Jun |
| Science China-Chemistry,2010, 53, 119-124. |
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| 2009 | Top |
|
|
| Construction of Multiring Frameworks by Metal-Free Cascade Reactions of Stable Isochromenylium Tetrafluoroborate |
| Hu Zhi-Long, Qian Wen-Jian, Wang Sheng, Wang Shaozhong, Yao Zhu-Jun |
| Journal of Organic Chemistry,2009, 22, 8787-8793. |
| 
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| Transformation of Reactive Isochromenylium Intermediates to Stable Salts and Their Cascade Reactions with Olefins |
| Hu Zhi-Long, Qian Wen-Jian, Wang Sheng, Wang Shaozhong, Yao Zhu-Jun |
| Organic Letters,2009, 11, 4676-4679. |
| 
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| Efficient Synthesis of 4-Amido-N(5)-acetyl-4-deoxyneuraminic Acid and Its Application to the C-4 Modification of Sialic Acids |
| Gao Zheng-Xi, Wang Meng, Wang Shaozhong, Yao Zhu-Jun |
| Organic Letters,2009, 11, 3678-3681. |
| 
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| Stereoselective Synthesis of the Functionalized C2-C10 Fragment of Clavulactone |
| Zhou Zuo-Zhong, Suo Dong, Yang Zhen-Yu, Chen Lin, Hu Tai-Shan, Yao Zhu-Jun |
| Chinese Journal of Chemistry,2009, 27, 135-140. |
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| 2008 | Top |
|
|
| Expeditious Total Syntheses of Camptothecin and 10-Hydroxycamptothecin |
| Liu Guan-Sai, Dong Qing-Li, Yao Yuan-Shan, Yao Zhu-Jun |
| Organic Letters,2008, 23, 5393-5396. |
| 
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|
|
| Development of New Pyrrolocoumarin Derivatives with Satisfactory Fluorescent Properties and Notably Large Stokes Shifts |
| Chen Lei, Hu Tai-Shan, Yao Zhu-Jun |
| European Journal of Organic Chemistry,2008, 36, 6175-6182. |
|
|
| Site-Specific Fluorescent Labeling Approaches for Naringenin, an Essential Flavonone in Plant Nitrogen-Fixation Signaling Pathways |
| Chen Lei, Li Fen-Qing, Hou Bi-He, Hong Glio-Fan, Yao Zhu-Jun |
| Journal of Organic Chemistry,2008, 73, 8279-8285. |
| 
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|
| Total synthesis of platensimycin: a review |
| Yao Yuan-Shan, Yao Zhu-Jun |
| Chinese Journal of Organic Chemistry,2008, 28, 1553-1560. |
|
|
| Biomimetic total syntheses of cassiarins A and B |
| Yao Yuan-Shan, Yao Zhu-Jun |
| Journal of Organic Chemistry,2008, 73, 5221-5225. |
| 
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|
| Synthesis of the biotinylated artemisinin derivative |
| Zhong Chun-Long, Yao Zhu-Jun |
| Acta Chimica Sinica,2008, 66, 1074-1078. |
|
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| Metal-free synthesis of alkynyl imines using an oxophosphonium-mediated approach at ambient temperatures |
| Dong Qing-Li, Liu Guan-Sai, Zhou Hai-Bin, Chen Lin, Yao Zhu-Jun |
| Tetrahedron Letters,2008, 10, 1636-1640. |
|
|
| Tuning the Acyclic Ether Moiety of Anticancer Agent AA005 with Conformationally Constrained Fragments |
| Liu Hai-Xia, Shao Fei, Li Gang-Qin, Xun Guo-Liang, Yao Zhu-Jun |
| Chemistry-A European Journal,2008, 14, 8632-8639. |
| 
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| 2007 | Top |
|
|
| Short and efficient total synthesis of luotonin a and 22-hydroxyacuminatine using a common cascade strategy |
| Zhou Hai-Bin, Liu Guan-Sai, Yao Zhu-Jun |
| Journal of Organic Chemistry,2007, 72, 6270-6272. |
| 
|
|
|
| An inexpensive fluorescent labeling protocol for bioactive natural products utilizing Cu(I)-catalyzed Huisgen reaction |
| Zhang Yan-Hong, Gao Zheng-Xi, Zhong Chun-Long, Zhou Hai-Bin, Chen Lei, Wu Wen-Min, Peng Xin-Jun, Yao Zhu-Jun |
| Tetrahedron,2007, 63, 6813-6821. |
| 
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| Annonaceous acetogenin mimics bearing a terminal lactam and their cytotoxicity against cancer cells |
| Liu Hai-Xia, Huang Guo-Rui, Zhang Huan-Ming, Wu Jia-Rui, Yao Zhu-Jun |
| Bioorganic & Medicinal Chemistry Letters,2007, 17, 3426-3430. |
| 
|
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|
| Total synthesis, assignment of absolute stereochemistry, and structural revision of chlorofusin |
| Qian Wen-Jian, Wei Wan-Guo, Zhang Yong-Xia, Yao Zhu-Jun |
| Journal of the American Chemical Society,2007, 129, 6400-6401. |
| 
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|
|
| Parallel synthesis of individual shikimic acid-like molecules using a mixture-operation strategy and ring-closing enyne metathesis |
| Hu Fang, Zhang Yan-Hong, Yao Zhu-Jun |
| Tetrahedron Letters,2007, 48, 3511-3515. |
| 
|
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|
| Highly efficient and mild cascade reactions triggered by bis(triphenyl)oxodiphosphonium trifluoromethanesulfonate and a concise total synthesis of camptothecin |
| Zhou Hai-Bin, Liu Guan-Sai, Yao Zhu-Jun |
| Organic Letters,2007, 9, 2003-2006. |
| 
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| 2006 | Top |
|
|
| An efficient synthesis of selective human NR2A antagonist NVP-AAM077 |
| Li Gang-Qin, Su Wei-Ke, Yao Zhu-Jun |
| Chinese Journal of Chemistry,2006, 24, 1784-1787. |
|
|
| A concise synthesis of L-3-(o-methoxybenzoyl)alanine, a selective kynurenine hydroxylase inhibitor |
| Ma Xiang-Dong, Yao Zhu-Jun |
| Acta Chimica Sinica,2006, 64, 2197-2200. |
|
|
| Bidirectional synthesis of the central amino acid of chloptosin |
| Hong Wen-Xu, Chen Ling-Jun, Zhong Chun-Long, Yao Zhu-Jun |
| Organic Letters,2006, 8, 4919-4922. |
| 
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|
|
| Ring-closing metathesis-based synthesis of (3R,4R,5S)-4-acetylamino-5-amino-3-hydroxycyclohex-1-ene-carboxylic acid ethyl ester: A functionalized cycloalkene skeleton of GS4104 |
| Cong Xin, Yao Zhu-Jun |
| Journal of Organic Chemistry,2006, 71, 5365-5368. |
| 
|
|
|
| Bromoetherification-based strategy towards the spirocyclic chromophore of chlorofusin |
| Wei Wan-Guo, Qian Wen-Jian, Zhang Yong-Xia, Yao Zhu-Jun |
| Tetrahedron Letters,2006, 47, 4171-4174. |
| 
|
|
|
| Application of a regioselective Mannich reaction on naringenin and its use in fluorescent labeling |
| Chen Lei, Hu Tai-Shan, Zhu Jing, Wu Houming, Yao Zhu-Jun |
| Synlett,2006, 8, 1225-1229. |
|
|
| Pauson-khand approach towards enantiopure C-2-symmetric polycyclic compound from D-mannitol |
| He Y.-T., Xue S., Yao Zhu-Jun |
| Acta Chimica Sinica,2006, 64, 169-174. |
|
|
| Studies on natural cryptophycins and their mimetics: A review |
| Zha H.-Y., Yao Zhu-Jun |
| Chinese Journal of Organic Chemistry,2006, 26, 27-42. |
|
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| 2005 | Top |
|
|
| Efficient construction of novel alpha-keto spiro ketal and the total synthesis of (+/-)-terreinol |
| Wei Wan-Guo, Zhang Y.-X., Yao Zhu-Jun |
| Tetrahedron,2005, 61, 11882-11886. |
| 
|
|
|
| Preparation of enantiomerically pure 2-(1 '-aminomethyl)furan derivatives and synthesis of an unnatural polyhydroxylated piperidine |
| Cong X., Liu K.-G., Liao J., Yao Zhu-Jun |
| Tetrahedron Letters,2005, 46, 8567-8571. |
| 
|
|
|
| An iterative acetylene-epoxide coupling strategy for the total synthesis of longimicin C |
| He Y.-T., Xue S., Hu T.-S., Yao Zhu-Jun |
| Tetrahedron Letters,2005, 46, 5393-5397. |
| 
|
|
|
| Synthesis studies toward chloroazaphilone and vinylogous gamma-pyridones: Two common natural product core structures |
| Wei Wan-Guo, Yao Zhu-Jun |
| Journal of Organic Chemistry,2005, 70, 4585-4590. |
| 
|
|
|
| Chemoselective deprotection of cyclic N,O-aminals using catalytic bismuth(III) bromide in acetonitrile |
| Cong X., Hu F., Liu K.-G., Liao Q.-J., Yao Zhu-Jun |
| Journal of Organic Chemistry,2005, 70, 4514-4516. |
| 
|
|
|
| Macrocyclization studies and total synthesis of cyclomarin C, an anti-inflammatory marine cyclopeptide |
| Wen S.-J., Hu T.-S., Yao Zhu-Jun |
| Tetrahedron,2005, 61, 4931-4938. |
| 
|
|
|
| Stereoselective synthesis of new modified conformationally constrained L-tyrosine analogue with potential applications to SH2 domain ligands |
| Liu F., Hu T.-S., Yao Zhu-Jun |
| Tetrahedron,2005, 61, 4971-4981. |
| 
|
|
|
| Synthesis of a tetra-deuterium-labeled derivative of potent and selective anticancer agent AA005 |
| Liu H.-X., Yao Zhu-Jun |
| Tetrahedron Letters,2005, 46, 3525-3528. |
| 
|
|
|
| Synthesis of two naturally occurring 4-hydroxylated butenolides with PTP1B inhibitory activity |
| Zhao Y., Jiang S., Guo Y.-W., Yao Zhu-Jun |
| Chinese Journal of Chemistry,2005, 23, 173-175. |
|
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| 2004 | Top |
|
|
| A chiron-based approach for the synthesis of tricyclic tyrosine analogue |
| Liu F., Jiao J., Zha H.-Y., Yao Zhu-Jun |
| Chinese Journal of Chemistry,2004, 22, 1022-1028. |
|
|
| RCM approaches toward the diastereoselective synthesis of vicinal trans-diaminocyclitols from L-serine |
| Cong X., Liao Q.-J., Yao Zhu-Jun |
| Journal of Organic Chemistry,2004, 69, 5314-5321. |
| 
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|
|
| Total synthesis of cyclomarin C |
| Wen S.-J., Yao Zhu-Jun |
| Organic Letters,2004, 6, 2721-2724. |
| 
|
|
|
| Synthesis of 4-azido-4-deoxy-Neu5,7,8,9Ac(4)2en1Me. A key intermediate for the synthesis of GG167 from D-glucono-delta-lactone |
| Liu K.-G., Yan S., Wu Y.-L., Yao Zhu-Jun |
| Organic Letters,2004, 6, 2269-2272. |
| 
|
|
|
| Synthesis of (2R,3aR,8aR)-6-chloro-3a-hydroxy-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indole-2-carboxylic acid methyl ester by reductive cyclization |
| Hong W.-X., Yao Zhu-Jun |
| Chinese Journal of Chemitry,2004, 22, 365-370. |
|
|
| Parallel fragment assembly strategy towards multiple-ether mimicry of anticancer annonaceous acetogenins |
| Jiang S., Li Y., Chen X.-G., Hu T.-S., Wu Y.-L., Yao Zhu-Jun |
| Angewandte Chemie-International Edition,2004, 43, 329-334. |
| 
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| 2003 | Top |
|
|
| Synthesis of a new stable conformationally constrained 2,7-anhydrosialic acid derivative |
| Liu K.-G., Zhou H.-B., Wu Y.-L., Yao Zhu-Jun |
| Journal of Organic Chemistry,2003, 68, 9528-9531. |
| 
|
|
|
| Studies on the synthesis of (2S,3R)-3-hydroxy-3-methylproline via C-2-N bond formation |
| Shen J.-W., Qin D.-G., Zhang H.-W., Yao Zhu-Jun |
| Journal of Organic Chemistry,2003, 68, 7479-7484. |
| 
|
|
|
| Synthesis of a new conformation-constrained L-tyrosine, analogue as a potential scaffold for SH2 domain ligands |
| Liu F., Zha H.-Y., Yao Zhu-Jun |
| Journal of Organic Chemistry,2003, 68, 6679-6684. |
| 
|
|
|
| A practical procedure for multisubstituted beta-naphthols and their derivatives |
| Wei W.-G., Yao Zhu-Jun |
| Tetrahedron,2003, 59, 6621-6625. |
| 
|
|
|
| An efficient enantioselective synthesis of the acyl side chain of polyoxypeptins |
| Qin D.-G., Yao Zhu-Jun |
| Tetrahedron Letters,2003, 44, 571-574. |
| 
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|
| 2002 | Top |
|
|
| Synthesis of a mimicking hybrid of Annonaceous acetogenin with steroid for antitumoral activity investigation |
| Jiang S., Wu Y.-L., Yao Zhu-Jun |
| Chinese Journal of Chemistry,2002, 20, 1393-1400. |
|
|
| Sharpless AD strategy toward the gamma-methyl butenolide unit of acetogenins: enantioselective synthesis of butenolide I and II with mosquito larvicidal activity |
| He Y.-T., Yang H.-N., Yao Zhu-Jun |
| Tetrahedron,2002, 58, 8805-8810. |
| 
|
|
|
| Recent progress of the synthetic study on sialic acid (N-acetylneuaminic acid) and its analogs |
| Li L.-S., Liu K.-G., Yao Zhu-Jun, Wu Yu-Lin |
| Chinese Journal of Organic Chemistry,2002, 22, 718-734. |
|
|
| A new synthesis of Neu5Ac from D-glucono-delta-lactone |
| Liu Ke-Gang, Yan Shi, Wu Yu-Lin, Yao Zhu-Jun |
| Journal of Organic Chemitry,2002, 67, 6758-6763. |
| 
|
|
|
| Synthesis of a fully protected (2S,3R)-N-(1 ',1 '-dimethyl-2 '-propenyl)-3-hydroxytryptophan from tryptophan |
| Wen S.-J., Zhang H.-W., Yao Zhu-Jun |
| Tetrahedron Letters,2002, 43, 5291-5294. |
| 
|
|
|
| First synthesis of mosquito larvicidal butenolides I and II |
| Jiang S., Wu Yu-Lin, Yao Zhu-Jun |
| Chinese Journal of Chemistry,2002, 20, 692-696. |
|
|
| Mimicry of annonaceous acetogenins: Enantioselective synthesis of a (4R)-hydroxy analogue having potent antitumor activity |
| Jiang Sheng, Liu Hai-Zhong, Sheng Gang, Zeng Bu-Bing, Cheng Xiao-Guang, Wu Yu-Lin, Yao Zhu-Jun |
| Journal of Organic Chemistry,2002, 67, 3404-3408. |
| 
|
|
|
| Enantioselective synthesis of (2S,3R)-3-hydroxy-3-methylproline, a novel amino acid found in polyoxypeptins |
| Qin Dong-Guang, Zha Hui-Yan, Yao Zhu-Jun |
| Journal of Organic Chemitry,2002, 67, 1038-1040. |
| 
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|
| Electronic effect of indolecarboxaldehyde in the condensation with t-butyl bromoacetate promoted by biazaborolidine |
| Wen S.-J., Yao Zhu-Jun |
| Acta Chimica Sinica,2002, 60, 129-133. |
|
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| Top |
| List of Publications before 2002 | 1. Wu,P., Chen,W.-S., Hu, T.-S., Yao, Z.-J., Wu, Y.-L. Annonaceous Acetogenin from Annona Atemoya Seeds. J. Asian Nat. Prod. Research2001, 3, 177. 2. Wu, Y.-L., Wu, W.-L., Yao, Z.-J., Li, Y.-L., Wang, Y.-F., Li, J.-C., Sun, X.-L., Peng, Z.-H., Yu, Q., Hu, T.-S., Zeng, B.-B., Wang, X.-Z. Syntheses of Enantiopure Natural Products from Sugars. Chinese J. Org. Chem. 2001, 21, 1051. 3. Atabey, N.; Gao, Y.;Yao, Z.-J.; Brechenridge, D.; Soon, L.; Burke Jr., T.R.; Bottaro, D.P. Potent blockade of hepatocyte growth factor-stimulated cell motility by selective inhibitors of Grb2-c-Met interaction. J. Biol. Chem. 2001, 276, 14308-14314. 4. Burke Jr., T. R., Yao, Z.-J., Ye, B., Miyoshi, K., Otaka, A., Wu., L., Zhang, Z.-Y. Phospho-azatyrosine, a less effective protein-tyrosine phosphatase substrate than phosphotyrosine. Bioorganic & Medicinal Chemistry Letters2001, 11, 1265-8. 5. Burke Jr.,T. R., Yao, Z.-J., Gao, Y., Wu, J. X., Zhu, X., Luo, J. H., Guo, R., Yang, D. N-Terminal Carboxyl and Tetrazole-Containing Amides as Adjuvants to Grb2 SH2 Domain Ligand Binding. Bioorg. Med. Chem.2001, 9, 1439-1445. 6. Burke Jr., T. R., Yao, Z.-J., Liu, D.-G., Voigt, J., Gao, Y. Phosphoryltyrosyl Mimetics in the Design of Peptide-Based Signal Transduction Inhibitors. Biopolymers2001, 60, 32-44. 7. Zhang, Y.-L., Yao, Z.-J., Sarmiento, M., Wu, L., Burke, Jr., T. R., Zhang, Z.-Y. Isothermal Titration Calorimetric Study of Ligand Binding to Protein-Tyrosine Phosphatase 1B and Its Substrate-Trapping Mutants. J. Biol. Chem.2000, 275(44), 34205-34212. 8. Long, Y.-Q., Lung, F.-D. T., Voigt, J. H., Yao, Z.-J., Burke, Jr., T. R., Yang, D., Luo, J. H., Guo, R., King, C. K., Roller, P. P. High affinity nonphosphorylated cyclic peptide inhibitors of Grb2-SH2 / growth factor receptor interactions. In Peptides: Frontier of Peptide Science, Proc. of 16th American Peptide Symposium, Tam, J. P., and Kaumaya, P. T. P. (Eds), ESCOM/Kluwer Acad. Publishers, Dordect, The Netherlands,2000, 568-570. 9. Yao, Z.-J., Barchi, J. J., Burke, Jr., T. R. Design and synthesis of a new tyrosine analogue having c1 and c2 angles constrained to values observed for an SH2 domain-bound phosphotyrosyl residue. In Peptides for the New Millennium: Proc. of 16th American Peptide Symposium, Fields, G. B., Tam, J. P., and Barany, G. (Eds), Kluwer Acad. Publishers, Dordect, The Netherlands,2000, p576-8. 10. Gao, Y., Yao, Z.-J., Voigt, J. H., Luo, J. H., Yang, D., Burke, Jr., T. R. Novel phosphotyrosyl mimetics for the preparation of potent small molecule Grb2 SH2 domain inhibitors. In Peptides for the New Millennium: Proc. of 16th American Peptide Symposium, Fields, G. B., Tam, J. P., and Barany, G. (Eds), Kluwer Acad. Publishers, Dordect, The Netherlands, 2000, p566-7. 11. Gao, Y., Luo, J., Yao, Z.-J., Guo, R., Zou, H., Kelley, J., Voigt, J. H., Yang, D., Burke, Jr., T. R. Inhibition of Grb2 SH2 Domain Binding by Non-Phosphate Containing Ligands 2. 4-(2-Malonyl)phenylalanine as a potent Phosphotyrosyl Mimetic. J. Med. Chem.2000,43, 911-920. 12. Burke Jr., T.R.; Gao, Y.; Yao, Z.-J.; Voigt, J.; Luo, J.; Dajun, Y. Potent non phosphate- containing Grb2 SH2 domain inhibitors. Peptide Chemistry 1999. Proceedings of the 36th Japanese Peptide Symposium, Ed. by N. Fujii,The Japanese Peptide Society, 2000, pp 49-52. 13. Yao, Z.-J., Wu, H.-P., Wu, Y.-L. Polyether Mimics of Natural Occurring Cytotoxic Annonaceous Acetogenins. J. Med. Chem.2000,43, 2484-2487. 14. Liu, D.-G.; Yao, Z.-J.;Gao, Y.; Burke, T.R., Jr. Large scale preparation of cell permeable, non-phosphate containing Grb2 SH2 domain inhibitors. Organic Preparations and Procedures International2000,32, 197-201. 15. Chen, H., Cong, L.-N., Li, Y., Yao, Z.-J., Wu, L., Zhang, Z.-Y., Burke Jr., T. R., Quon, M. J. A Phosphotyrosyl Mimetic Peptide Reverses Impairment of Insulin-stimulated Translocation of Glut4 Caused by Overexpression of PTP1B in Rat Adipose Cells. Biochemistry1999, 38(1), 384-389. 16. Yao, Z.-J., King, C. R., Cao, T., Kelley, J., Milne, G. W. A., Voigt, J. H., Burke Jr., T. R. Potent Inhibition of Grb2 SH2, Domain Binding by Non-Phosphate Cotaining Ligands. J. Med. Chem.1999,42(1), 25-35. 17. Burke Jr., T. R., Luo, J., Yao, Z.-J., Gao, Y., Milne, G. W. A., Voigt, J. H., King, C. R., Yang, D. Monocarboxylic-Based Phosphotyrosyl Mimetics in the Design of Grb2 SH2 Domain Inhibitors. Bioorganic and Medicinal Chemistry Lett. 1999,9, 347-352. 18. Yao, Z.-J., Gao, Y., Voigt, J. H., Ford, Jr., H., Burke Jr., T. R. Synthesis of Fmoc-Protected 4-Carboxydifluoromethyl-L-phenylalanine: A Phosphotyrosyl Mimetic of Potential Use for Signal Transduction Studies. Tetrahedron.1999,55, 2865-2874. 19. Yu, Q., Yao, Z.-J., Chen, X.-G., Wu, Y.-L. Total Synthesis of (10R) and (10S)-corossolin, Determination of the C-10 configuration and the Unexpected Differential Toxicity toward Cancer Cell Caused by the Configuration at C-10. J. Org. Chem.1999, 64, 2440-2445. 20. Long, Y.-Q., Yao, Z.-J., Lung, F.-D. T., Voigt, J. H., King, C. R., Burke, Jr., T. R., Roller, P. P. Overlapping function of amino acids in position-2 and Y0 leading to high affinity nonphosphorylated peptide ligands of Grb2-SH2 domain. Biochem. Biphys. Res. Comm.1999, 264, 902-908. 21. Yao, Z.-J., Gao, Y., Burke, T. R., Jr. Preparation of L-N-Fmoc-Pmp(tBu2)-OH From L-Tyrosine. Tetrahedron: Asymmetry 1999, 10, 3727-3734. 22. Wu, Y.-L., Chen, H.-B., Jiang, K., Li, Y., Shan, F., Wang, D.-Y., Wang, Y.-F., Wu, W.-M., Wu, Y., Yao, Z.-J., Yue, Z.-Y., Zhou, C.-M. Interaction of biomolecules with qinghaosu (artemisinin) and its derivatives in the presence of ferrous ion – an exploration of antimalarial mechanism. Pure Appl. Chem.1999, 71, 1139-1142. 23. Burke, T. 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Synthesis of annonaceous acetogenin (4S, 5S) and (4S, 5R)-muricatacin as well as confirmation of absolute configuration of the tetrahydrofuran segment of annonacin. Acta Chim. Sinica1992, 50, 901. | Top |
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CCS Chem. 2021, 3, 664–677.(DOI: org/10.31635/ccschem.021.202000691)
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