The Yao Group


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View by Year:2017, 2016, 2015, 2014,  20132012  2011201020092008200720062005200420032002, before 2002

2017

Top

Azepinoindole Synthesis via a N‑Bromosuccinimide-Induced Cycloisomerization of Enaminoester/Enaminone
Lina Chang, Tao Guo, Ziyi Wang, Shaozhong Wang,and Zhu-Jun Yao
J. Org. Chem. 2017, 82, 1567−1574 (DOI: 10.1021/acs.joc.6b02760)

Nodupetide, a potent insecticide and antimicrobial from Nodulisporium sp. associated with Riptortus pedestris
Hui Min Wu, Li Ping Lin, Qin Lan Xu, Wen Bo Han, Song Zhang, Ze Wen Liu, Ya Ning Mei,Zhu Jun Yao,and Ren Xiang Tan
Tetrahedron Letters. 2017, 58, 663C665DOI.org/10.1016/j.tetlet.2017.01.009

2016

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Michael addition-based cyclization strategy in the total synthesis of Lycopodium alkaloids
Lin-Rui Zhong and Yao Zhu-Jun*
SCIENCE CHINA Chemistry. 2016. 59. 1079-1087 (DOI:10.1007/s11426-016-0056-0)

Gram-Scale Laboratory Synthesis of UM171, a Potent Agonist of Human Hematopoietic Stem Cell Self-Renewal
Sajjad Ali, Shun-Ming Yu, and Zhu-Jun Yao*
J. Org. Chem. 2016, 81, 10236−10241 (DOI:10.1021/acs.joc.6b01094)

Aerobic a-hydroxylation of b-keto esters and amides by co-catalysis of SmI3 and I2 under mild base-free conditions
Shun-Ming Yu, Kai Cui, Fei Lv , Zhen-Yu Yang*, Zhu-Jun Yao*
 Tetrahedron. Letters. 2016. 57. 2818-2821 (DOI:10.1016/j.tetlet.2016.05.052)

Convenient One-Step Synthesis of Benzo[c]phenanthridines by Three-Component Reactions of Isochromenylium Tetrafluoroborates and Stilbenes in Acetonitrile
Gang-Gang ChenJun-Qiang WeiXiaoliang Yang*, and Zhu-Jun Yao*
Org. Lett. 2016, 18, 1502C1505 (DOI: 10.1021/acs.orglett.6b00010)

Enantioselective Total Synthesis of Lycoposerramine-Z Using Chiral Phosphoric Acid Catalyzed Intramolecular Michael Addition

Lan-De ZhangLin-Rui ZhongJie XiXiao-Liang Yang*, and Zhu-Jun Yao*
J. Org. Chem. 2016, 81, 1899C1904 (DOI: 10.1021/acs.joc.5b02723)

2015

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Kinetic or Dynamic Control on a Bifurcating Potential Energy Surface?An Experimental and DFT Study of Gold-Catalyzed Ring Expansion and Spirocyclization of 2-Propargyl--tetrahydrocarbolines
Zhang Lei,Yi Wang,Yao Zhu-Jun,Wang Shao-Zhong,Yu Zhi-Xing
J. Am. Chem. Soc. 2015, 137, 13290C13300(DOI:10.1021/jacs.5b05971)

Synthesis of Tricyclo[4,3,1,01,5]decane Core of Plumisclerin A Using PausonCKhand Annulation and SmI2-Mediated Radical Cyclization

Chen Ji-Peng,He Wei,Yang Zhen-Yu,and Yao Zhu-Jun
Org. Lett. 2015, 17, 3379C3381(DOI:10.1021/acs.orglett.5b01563)

Efficient Synthesis of Octahydrophenanthrene Derivatives with Mild Cascade Reactions of Isochromenylium Tetrafluoroborates and Bifunctional Styrenes ,
Mo Lei, Wu Lin-Lin,  Wang Shao-Zhong, Yao Zhu-Jun
Org. Lett. 2015, 17, 3314C3317(DOI:10.1021/acs.orglett.5b01532)

 
The last and next decades of the Asian Core Program on cutting-edge organic chemistry in Asia
Minoru Isobe, Atsushi Nishida, Yeun-Mun Choo, Noorsaadah Abd. Rahman, Poonsakdi Ploypradith, Somsak Ruchirawat, Guo-Qiang Lin, Ang Li, Zhu-Jun Yao, Biing-Jiun Uang, Chun-Chen Liao, Pauline Chiu, Byeong Moon Kim, Teck Peng Loh
Chemistry - An Asian Journal. 2015, 10, 790-804


Annonaceous acetogenin mimic AA005 induces cancer cell death via apoptosis inducing factor through a caspase-3-independent mechanism
Han Bing, Wang Tong-Dan, Shen Shao-Ming, Yu Yun, Mao Chan, Yao Zhu-Jun, Wang Li-Shun
BMC Cancer  2015, 15, 139


Short Protecting Group-free Syntheses of Camptothecin and 10-Hydroxycamptothecin Using Cascade Methodologies
Xu Peng, Chen Dong-Sheng Chen, Xi Jie, Yao Zhu-Jun
Chemistry - An Asian Journal. 2015, 10, 976-981


Stereodivergent total synthesis of chlorofusin and its all seven chromophore diastereomers
Qiu Hai-Bo, Qian Wen-Jian, Yu Shun-Ming, Yao Zhu-Jun

Tetrahedron 2015, 71, 370-380

2014

Top


Total Synthesis of Ascididemin-Type Alkaloids Using Alkyne Building Blocks
Yin Hao, Shan Naiyu, Wang Shaozhong, Yao Zhu-Jun
Journal of Organic Chemistry . 2014, 79, 9748-9753


Total synthesis of proposed structure of coibamide A, a highly N- and O-methylated cytotoxic marine cyclodepsipeptide
He Wei, Qiu Hai-Bo, Chen Yi-Jie, Xi Jie, Yao Zhu-Jun
Tetrahedron Letters. 2014, 55, 6109-6112


Unified flexible total synthesis of chlorofusin and artificial Click mimics as antagonists against p53CHDM2 interactions
Qiu Hai-Bo, Chen Xin-Ya, Li Qing, Qian Wen-Jian, Yu Shun-Ming, Tang Gong-Li, Yao Zhu-Jun
Tetrahedron Letters. 2014, 55, 6055-6059


Total Syntheses of Lycoposerramine-V and 5-epi-Lycoposerramine-V
Zhang Lan-De, Zhou Ting-Ting, Qi Sen-Xing, Xi Jie, Yang Xiao-Liang, Yao Zhu-Jun
Chemistry - An Asian Journal. 2014, 9, 2740-2744


Asymmetric Annulation of 3‑Alkynylacrylaldehydes with Styrene-Type Olefins by Synergetic Relay Catalysis from AgOAc and Chiral Phosphoric Acid
Zhang Hao, Zhu Le, Wang Shaozhong, Yao Zhu-Jun
Journal of Organic Chemistry, 2014, 79, 7063-7074


Regio-controlled synthesis of unsymmetrical pyrazine-fused sinomenine derivatives and discriminate substitution effects on TNF- inhibitory activity
Zhou Tingting, Hou Jian, Wang Meng, Ma Liyan, Wu Linlin, Wang Shaozhong, Sun Bing, Yao Zhu-Jun
Tetrahedron 2014. 70. 5475-5482


New cytotoxic annonaceous acetogenin mimetics having a nitrogen-heterocyclic terminal and their application to cell imaging
Chen Yi-Jie, Jin Sheng, Xi Jie, Yao Zhu-Jun
Tetrahedron 2014. 70. 4921-4928


Total synthesis of ent-(−)-azonazine using a biomimetic direct oxidative cyclization and structural reassignment of natural product
Zhao Ji-Chen,Yu Shun-Ming,Qiu Hai-Bo,Yao Zhu-Jun
Tetrahedron. 2014. 70. 3197C3210


Biological evaluation of new mimetics of annonaceous acetogenins: Alteration of right scaffold by click linkage with aromatic functionalities
Liu Yanghan, Xiao Qicai, Liu Yongqiang, Li Zheng, Qiu Yatao, Zhou Guang-Biao, Yao Zhu-Jun, Jiang Sheng
 European Journal of Medicinal Chemistry. 2014. 78. 248-258


Identification of novel bivalent mimetics of annonaceous acetogenins via a scaffold-hopping strategy
Liu Yanghan, Liu Yongqiang, Li Zhen, Zhou Guang-Biao, Yao Zhu-Jun, Jiang Sheng
Bioorganic & Medicinal Chemistry Letters.  2014. 24. 1650-1653


Azocinoindole Synthesis by a Gold(I)-Catalyzed Ring Expansion of 2-Propargyl-b-Tetrahydrocarboline
Zhang Lei, Chang Lina, Hu Hongwen, Wang Huaqin, Yao Zhu-Jun, Wang Shaozhong
Chemistry - A European Journal. 2014, 20, 2925-2932


2013

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Assembly of indolo[1,2-c]quinazolines using ZnBr2-promoted domino hydroaminationCcyclization
Xu Min, Xu Ke, Wang Shaozhong, Yao Zhu-Jun
Tetrahedron Letters, 2013, 54, 4675-4678


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Chinese Science Bulletin, 2013, 58, 2872-2885

Synthesis of 2-vinyl-2H-benzotriazoles via NIS-promoted regio/stereoselective addition of 1H-benzotriazole to alkynes
Zhang ZhenHua, Chang Lina, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun
RSC Advances, 2013, 3, 18446-18452


Biomimetic Synthesis of ent-(−)-Azonazine and Stereochemical Reassignment of Natural Product
Zhao Ji-Chen, Yu Shun-Ming, Liu Yun, Yao Zhu-Jun
Organic Letters, 2013, 15, 4300-4303


Asymmetric Cascade Annulation Based on Enantioselective OxaDiels−Alder Cycloaddition of in Situ Generated Isochromenyliums by Cooperative Binary Catalysis of Pd(OAc)2 and (S)‑Trip
Yu Shu-Yan, Zhang Hao, Gao Yang, Mo Lei, Wang Shaozhong,  Yao Zhu-Jun
Journal of the American Chemical Society,  2013, 135, 11402-11407


Asymmetric Michael addition of 4H-thiopyran-4-one to nitroolefins catalyzed by diamine mono-N-sulfonamide and its application to concise synthesis of enantiopure multiring heterocycles
Mo Lei, Tang Huang,  Yao Zhu-Jun
Tetrahedron, 2013, 69, 6897-6905


Dual-Functional abeo-Taxane Derivatives Destabilizing Microtubule Equilibrium and Inhibiting NF-B Activation
Yu Zhao, Jia Su, Masuo Goto, Susan L. Morris-Natschke, Yan Li, Qin-Shi Zhao, Zhu-Jun Yao, Kuo-Hsiung Lee
Journal of Medicinal Chemistry, 2013, 56, 4749−4757


Asymmetric One-Pot Sequential Mannich/Hydroamination Reaction by Organo- and Gold Catalysts: Synthesis of Spiro[pyrrolidin-3,2-oxindole] Derivatives
Chen Xianjie, Chen Hui, Ji Xun, Jiang Hualiang, Yao Zhu-Jun, Liu Hong
Organic Letters, 2013, 15, 1846C1849


Organocatalytic enantioselective conjugate addition of 2-nitrocyclohexanone to acrylaldehyde: a concise two-step synthesis of chiral building block 1-azaspiro[4.5]decan-6-one

Ding Xiao-Hua, Cui Wei-Chen, Li Xiang, Ju Xuan, Liu Dan, Wang Shaozhong, Yao Zhu-Jun
Tetrahedron Letters, 2013, 54, 1956-1959


Assembly of fused indenes via Au(I)-catalyzed C1CC5 cyclization of enediynes bearing an internal nucleophile
Hou Qiwen, Zhang Zhenhua, Kong Fanji, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun
Chemical Communications, 2013, 49, 695-697.


2012

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Sinomenine derivatives with embedment of nitrogen-containing heterocycles exhibiting potent TNF-inhibitory activity
Wang Meng, Ma Li-Yan, Lou Yang-Tong, Bian Chao, Zhou Ting-Ting, Zhou Hai-Bin, Liao Hong-Ze, Ma Zhao, Yin Dong-Sheng, Wang Shaozhong, Yang Zhen-Yu, Sun Bing, Yao Zhu-Jun
Science China Chemistry, 2012, 55, 2537-2547.

Assembly of pentacyclic pyrido[4,3,2-mn]acridin-8-ones via a domino reaction initiated by Au(I)-catalyzed 6-endo-dig cycloisomerization of N-propargylaminoquinones
Yin Hao, Kong Fanji, Wang Shaozhong, Yao Zhu-Jun
Tetrahedron Letters, 2012, 53, 7078-7082.


Gefitinib Analogue V1801 Induces Apoptosis of T790M EGFR-Harboring Lung Cancer Cells by Up-Regulation of the BH-3 Only Protein Noxa
Zhang Bo, Jiao Jiao, Liu Ying, Guo Liang-Xia, Zhou Bo, Li Gang-Qin, Yao Zhu-Jun, Zhou Guang-Biao
PLOS ONE, 2012, 7(11), e48748.

Identification of an Annonaceous Acetogenin Mimetic, AA005, as an AMPK Activator and Autophagy Inducer in Colon Cancer Cells
Liu Yong-Qiang, Cheng Xin, Guo Liang-Xia, Mao Chan, Chen Yi-Jie, Liu Hai-Xia, Xiao Qi-Cai, Jiang Sheng, Yao Zhu-Jun, Zhou Guang-Biao
PLOS ONE, 2012, 7(10), e47049.

Highly Enantioselective Michael Addition of 2-Oxindole- 3-carboxylate Esters to Nitroolefins Promoted by Cinchona Alkaloid-Thiourea-Brønsted Acid Cocatalysts
Chen Xian-Jie, Zhu Wei, Qian Wangke, Feng Enguang, Zhou Yu, Wang Jinfang, Jiang Hualiang, Yao Zhu-Jun, Liu Hong
Advanced Synthesis & Catalysis, 2012, 354, 2151-2156.


Protecting Group-Free Total Synthesis of (−)-Lannotinidine B
Ge Hui-Ming, Zhang Lan-De, Tan Ren-Xiang, Yao Zhu-Jun
Journal of the American Chemical Society, 2012, 134, 12323-12325.


Effect of Annonaceous Acetogenin Mimic AA005 on Proliferative Inhibition of Leukemia Cells in vitro and Its Possible Mechanisms
Han Bing, Yao Zhu-Jun, Wang Li-Shun
Journal of Experimental Hematology, 2012, 20, 549-553.


Enantioselective Total Synthesis of Marine Diterpenoid Clavulactone
Yang Zhen-Yu, Liao Hong-Ze, Shen Kang, Chen Yong-Fei, Yao Zhu-Jun
Angewandte Chemie International Edition, 2012, 51, 6484-6487.


Target-oriented multifunctional organocatalysis for enantioselective synthesis of bicyclo[3.3.1]nona-2,6-dien-9-ones. A formal asymmetric synthesis of huperzine A
Ding Xiao-Hua, Li Xiang, Liu Dan, Cui Wei-Chen, Ju Xuan, Wang Shaozhong, Yao Zhu-Jun
Tetrahedron, 2012, 68, 6240-6248.


A simple selective protocol for continuous two-stage fluorescent sensing of both MeHg+ and anti-MeHg+ agents in living cells
Mei De-Sheng, He Bao-Kun, Chen Lei, Yao Zhu-Jun
Tetrahedron Letters, 2012, 53, 3463-3466.


Brönsted acid-promoted dimerization of o-alkynylbenzaldehydes: a one-step synthesis of functionalized Kagans ether analogues
Zhang Hao, Cui Wei-Chen, Hu Zhi-Long, Yu Shu-Yan, Wang Shaozhong, Yao Zhu-Jun
RSC Advances, 2012, 2, 5101-5104.


Electronically unfavorable addition of electron-deficient olefins to isochromenylium tetrafluoroborates initiated by C-1 O-glycosylation
Yu Shu-Yan, Hu Zhi-Long, Zhang Hao, Wang Shaozhong, Yao Zhu-Jun
Tetrahedron Letters, 2012, 53, 2765-2768.


Regio- and stereoselective C10¨CH functionalization of sinomenine: an access to more potent immunomodulating derivatives
Lou Yang-Tong, Ma Li-Yan, Wang Meng, Yin Dongsheng, Zhou Ting-Ting, Chen Ai-Zhong, Ma Zhao, Bian Chao, Wang Shaozhong, Yang Zhen-Yu, Sun Bing, Yao Zhu-Jun
Tetrahedron, 2012, 68, 2172-2178.


Concise synthesis of zanamivir and its C4-thiocarbamido derivatives utilizing a [3+2]-cycloadduct derived from d-glucono--lactone
Zhu Xue-Bin, Wang Meng, Wang Shaozhong, Yao Zhu-Jun
Tetrahedron, 2012, 68, 2041-2044.

2011

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Development of Novel Conformation-Constrained Cytotoxic Derivatives of Cheliensisin A by Embedment of Small Heterocycles
Deng Xu, Su Jia, Zhao Yu, Peng Li-Yan, Yao Zhu-Jun, Zhao Qin-Shi
European Journal of Medicinal Chemistry, 2011, 46, 4238-4244.


Total Synthesis of 7-Ethyl-10-hydroxycamptothecin (SN38) and its Application to the Development of C18-Functionalized Camptothecin Derivativesivatives
Yao Yuan-Shan, Liu Jia-Li, Xi Jie, Miu Bukeyan, Liu Guan-Sai, Wang Shaozhong, Meng Linghua, Yao Zhu-Jun
Chemistry- A European Journal, 2011, 17, 10462-10469.


Modular assembly of cytotoxic acetogenin mimetics by click linkage with nitrogen functionalities
Mao Chan, Han Bing, Wang Li-Shan, Wang Shaozhong, Yao Zhu-Jun
MedChemComm, 2011, 2, 918-922.


CuCl(2)-Promoted 6-endo-dig Chlorocyclization and Oxidative Aromatization Cascade: Efficient Construction of 1-Azaanthraquinones from N-Propargylaminoquinones
Fei Na, Yin Hao, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun
Organic Letters, 2011, 13, 4208-4211.


Efficient synthesis of furoquinolinones using Hendrickson reagent-initiated cascade annulation
Xu Peng, Liu Guan-Sai, Xi Jie, Wang Shaozhong, Yao Zhu-Jun
Tetrahedron, 2011, 67, 5455-5460.


Generation of trans-arachidonic acid under nitrative stress is associated with upregulation of thromponsdin-1 in diabetic rats
Xu Lin, Liu Yu-Min, Yao Zhu-Jun, Xun Guo-Liang, Yu Wen-Juan, Liu Kun, Sun Xiao-Dong, Qiu Yun-Ping, Wu Hai-Xiang, Xu Xun
Chinese Medical Journal, 2011, 124, 1885-1889.

Evaluation of nitrative stress on retinal capillary by detection of trans-arachidonic acid with GC/MS in diabetic rats
Xu Lin, Xun Guo-Liang, Yao Zhu-Jun, Liu Yu-Min, Fan Ying, Sun Tao, Xu Xun
Chinese Journal of Experimental Ophthalmology, 2011, 29, 432-436.

Design, synthesis of symmetrical bivalent analogues mimetics of annonaceous acetogenins and their cytotoxicities
Xiao Qi-Cai, Liu Yong-Qiang, Qiu Ya-Tao, Yao Zhi-Yi, Zhou Guang-Biao, Yao Zhu-Jun, Jiang Sheng
Bioorganic & Medicinal Chemistry Letters, 2011, 21, 3613-3615.


Study on Iron-Catalyzed Oxidative Free Radical Dimerization of Isochromenylium Tetrafluoroborate
Song Xiao-Nan, Mo Lei, Hu Zhi-Long, Yang Zhen-Yu, Yao Zhu-Jun
Acta Chimica Sinica, 2011, 69, 680-686.

Syntheses and characterizations of novel pyrrolocoumarin probes for SNAP-tag labeling technology
Mei De-Sheng, Qu Yi, He Jin-Xiang, Chen Lei, Yao Zhu-Jun
Tetrahedron, 2011, 67, 2251-2259.


Facile Assembly of 11H-Indolo[3,2-c]quinoline by a Two-Step Protocol Involving a Regioselective 6-endo-Cyclization Promoted by the Hendrickson Reagent
Xu Min, Hou Qiwen, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun
Synthesis-Stuttgart, 2011, 4, 626-634.

Potent Antitumor Mimetics of Annonaceous Acetogenins Embedded with an Aromatic Moiety in the Left Hydrocarbon Chain Part
Xiao Qi-Cai, Liu Yong-Qiang, Qiu Ya-Tao, Zhou Guang-Biao, Mao Chan, Li Zheng, Yao Zhu-Jun, Jiang Sheng
Journal of Medicinal Chemistry, 2011, 54, 525-533.


Fragmentations of 13-oxo-taxyunnansin A and their application to preparation of abeo-paclitaxel and abeo-docetaxel analogues
Zhao Yu, Zhang Hong-Bin, Liu Ji-Kai, Su Jia, Li Yan, Yao Zhu-Jun, Zhao Qin-Shi
Tetrahedron Letters, 2011, 52, 139-142.


Three-Component Reactions of Isochromenylium Tetrafluoroborates via Non-Classical [4+2]-Intermediates: Mild One-Step Metal-Free Synthesis of Functionalized Dihydronaphthalenes and Tetrahydronaphthalenes
Hu Zhi-Long, Yang Zhen-Yu, Wang Shaozhong, Yao Zhu-Jun
Chemistry-A European Journal, 2011, 17, 1268-1274.


2010

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Synthesis of Tetrahydroisoquinolines via Cascade Reductive Amination of Isochromenylium Tetrafluoroborate with Primary Amines
Liao Hong-Ze, Hu Zhi-Long, Cui Kai, Jiao Jiao, Qin Yong, Yao Zhu-Jun
Synthesis-Stuttgart, 2010, 20, 3474-3480.

Efficient Synthesis of Phenanthridines Using Hendrickson Reagent Initiated Cascade Reaction under Mild Conditions
Xi Jie, Dong Qing-Li, Liu Guan-Sai, Wang Shaozhong, Chen Lin, Yao Zhu-Jun
Synlett, 2010, 11, 1674-1678.

Efficient Synthesis of Phenanthridines Using Hendrickson Reagent Initiated Cascade Reaction under Mild Conditions
Jiang Chun-Hui, Xu Min, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun
Journal of Organic Chemistry, 2010, 75, 4323-4325.


Synthesis of the cyclic nonapeptide of chlorofusin using a convergent [3+3+3]-fragment coupling strategy
Wang Yan-Li, Qian Wen-Jian, Wei Wan-Guo, Zhang Yue, Yao Zhu-Jun
Tetrahedron, 2010, 66, 3427-3432.


Short asymmetric synthesis of (S,S)-PDP using L-prolinol derivative as economic starting material
Song Xiao-Nan, Yao Zhu-Jun
Tetrahedron, 2010, 66, 2589-2593.


Direct nucleophilic C-1 addition of stable isochromenylium tetrafluoroborates under catalyst-free conditions: A new access to 1H-isochromenes
Hu Zhi-Long, Qian Wen-Jian, Yao Zhu-Jun
Science China-Chemistry, 2010, 53, 869-876.

Total Synthesis of Chloptosin, a Potent Apoptosis-Inducing Cyclopeptide
Yu Shun-Ming, Hong Wen-Xu, Wu Yuan, Zhong Chun-Long, Yao Zhu-Jun
Organic Letters, 2010, 12, 1124-1127.


Modification of poorly bioactive sinomenine into more potent immunosuppressive agents by embedding of drug-like fragments
Lou Yang-Tong, Zhou Hai-Bin, Zou Jia, Yan Ling-Chen, Bi En-Guan, Sun Bing, Yao Zhu-Jun
Tetrahedron Letters, 2010, 51, 485-488.


Azaanthraquinone assembly from N-propargylamino quinone via iodine-induced 6-endo-dig electrophilic cyclization
Fei Na, Hou Qi-Wen, Wang Shaozhong, Wang Huaqin, Yao Zhu-Jun
Organic & Biomolecular Chemistry, 2010, 8, 4096-4103.


Efficient Total Synthesis of (S)-14-Azacamptothecin
Liu Guan-Sai, Yao Yuan-Shan, Xu Peng, Wang Shaozhong, Yao Zhu-Jun
Chemistry-An Asian Journal, 2010, 5, 1382-1388.


Synthesis of N(11)-anchoring biotinylated artemisinin derivatives and their preliminary biological assessment
Pan Qi-Yu, Wang Shaozhong, Lu JinJian, Meng Linghua, Yao Zhu-Jun
Science China-Chemistry, 2010, 53, 119-124.

2009

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Construction of Multiring Frameworks by Metal-Free Cascade Reactions of Stable Isochromenylium Tetrafluoroborate
Hu Zhi-Long, Qian Wen-Jian, Wang Sheng, Wang Shaozhong, Yao Zhu-Jun
Journal of Organic Chemistry, 2009, 22, 8787-8793.


Transformation of Reactive Isochromenylium Intermediates to Stable Salts and Their Cascade Reactions with Olefins
Hu Zhi-Long, Qian Wen-Jian, Wang Sheng, Wang Shaozhong, Yao Zhu-Jun
Organic Letters, 2009, 11, 4676-4679.


Efficient Synthesis of 4-Amido-N(5)-acetyl-4-deoxyneuraminic Acid and Its Application to the C-4 Modification of Sialic Acids
Gao Zheng-Xi, Wang Meng, Wang Shaozhong, Yao Zhu-Jun
Organic Letters, 2009, 11, 3678-3681.


Stereoselective Synthesis of the Functionalized C2-C10 Fragment of Clavulactone
Zhou Zuo-Zhong, Suo Dong, Yang Zhen-Yu, Chen Lin, Hu Tai-Shan, Yao Zhu-Jun
Chinese Journal of Chemistry, 2009, 27, 135-140.

2008

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Expeditious Total Syntheses of Camptothecin and 10-Hydroxycamptothecin
Liu Guan-Sai, Dong Qing-Li, Yao Yuan-Shan, Yao Zhu-Jun
Organic Letters, 2008, 23, 5393-5396.


Development of New Pyrrolocoumarin Derivatives with Satisfactory Fluorescent Properties and Notably Large Stokes Shifts
Chen Lei, Hu Tai-Shan, Yao Zhu-Jun
European Journal of Organic Chemistry, 2008, 36, 6175-6182.

Site-Specific Fluorescent Labeling Approaches for Naringenin, an Essential Flavonone in Plant Nitrogen-Fixation Signaling Pathways
Chen Lei, Li Fen-Qing, Hou Bi-He, Hong Glio-Fan, Yao Zhu-Jun
Journal of Organic Chemistry, 2008, 73, 8279-8285.


Total synthesis of platensimycin: a review
Yao Yuan-Shan, Yao Zhu-Jun
Chinese Journal of Organic Chemistry, 2008, 28, 1553-1560.

Biomimetic total syntheses of cassiarins A and B
Yao Yuan-Shan, Yao Zhu-Jun
Journal of Organic Chemistry, 2008, 73, 5221-5225.


Synthesis of the biotinylated artemisinin derivative
Zhong Chun-Long, Yao Zhu-Jun
Acta Chimica Sinica, 2008, 66, 1074-1078.

Metal-free synthesis of alkynyl imines using an oxophosphonium-mediated approach at ambient temperatures
Dong Qing-Li, Liu Guan-Sai, Zhou Hai-Bin, Chen Lin, Yao Zhu-Jun
Tetrahedron Letters, 2008, 10, 1636-1640.

Tuning the Acyclic Ether Moiety of Anticancer Agent AA005 with Conformationally Constrained Fragments
Liu Hai-Xia, Shao Fei, Li Gang-Qin, Xun Guo-Liang, Yao Zhu-Jun
Chemistry-A European Journal, 2008, 14, 8632-8639.


2007

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Short and efficient total synthesis of luotonin a and 22-hydroxyacuminatine using a common cascade strategy
Zhou Hai-Bin, Liu Guan-Sai, Yao Zhu-Jun
Journal of Organic Chemistry, 2007, 72, 6270-6272.


An inexpensive fluorescent labeling protocol for bioactive natural products utilizing Cu(I)-catalyzed Huisgen reaction
Zhang Yan-Hong, Gao Zheng-Xi, Zhong Chun-Long, Zhou Hai-Bin, Chen Lei, Wu Wen-Min, Peng Xin-Jun, Yao Zhu-Jun
Tetrahedron, 2007, 63, 6813-6821.


Annonaceous acetogenin mimics bearing a terminal lactam and their cytotoxicity against cancer cells
Liu Hai-Xia, Huang Guo-Rui, Zhang Huan-Ming, Wu Jia-Rui, Yao Zhu-Jun
Bioorganic & Medicinal Chemistry Letters, 2007, 17, 3426-3430.


Total synthesis, assignment of absolute stereochemistry, and structural revision of chlorofusin
Qian Wen-Jian, Wei Wan-Guo, Zhang Yong-Xia, Yao Zhu-Jun
Journal of the American Chemical Society, 2007, 129, 6400-6401.


Parallel synthesis of individual shikimic acid-like molecules using a mixture-operation strategy and ring-closing enyne metathesis
Hu Fang, Zhang Yan-Hong, Yao Zhu-Jun
Tetrahedron Letters, 2007, 48, 3511-3515.


Highly efficient and mild cascade reactions triggered by bis(triphenyl)oxodiphosphonium trifluoromethanesulfonate and a concise total synthesis of camptothecin
Zhou Hai-Bin, Liu Guan-Sai, Yao Zhu-Jun
Organic Letters, 2007, 9, 2003-2006.


2006

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An efficient synthesis of selective human NR2A antagonist NVP-AAM077
Li Gang-Qin, Su Wei-Ke, Yao Zhu-Jun
Chinese Journal of Chemistry, 2006, 24, 1784-1787.

A concise synthesis of L-3-(o-methoxybenzoyl)alanine, a selective kynurenine hydroxylase inhibitor
Ma Xiang-Dong, Yao Zhu-Jun
Acta Chimica Sinica, 2006, 64, 2197-2200.

Bidirectional synthesis of the central amino acid of chloptosin
Hong Wen-Xu, Chen Ling-Jun, Zhong Chun-Long, Yao Zhu-Jun
Organic Letters, 2006, 8, 4919-4922.


Ring-closing metathesis-based synthesis of (3R,4R,5S)-4-acetylamino-5-amino-3-hydroxycyclohex-1-ene-carboxylic acid ethyl ester: A functionalized cycloalkene skeleton of GS4104
Cong Xin, Yao Zhu-Jun
Journal of Organic Chemistry, 2006, 71, 5365-5368.


Bromoetherification-based strategy towards the spirocyclic chromophore of chlorofusin
Wei Wan-Guo, Qian Wen-Jian, Zhang Yong-Xia, Yao Zhu-Jun
Tetrahedron Letters, 2006, 47, 4171-4174.


Application of a regioselective Mannich reaction on naringenin and its use in fluorescent labeling
Chen Lei, Hu Tai-Shan, Zhu Jing, Wu Houming, Yao Zhu-Jun
Synlett, 2006, 8, 1225-1229.

Pauson-khand approach towards enantiopure C-2-symmetric polycyclic compound from D-mannitol
He Y.-T., Xue S., Yao Zhu-Jun
Acta Chimica Sinica, 2006, 64, 169-174.

Studies on natural cryptophycins and their mimetics: A review
Zha H.-Y., Yao Zhu-Jun
Chinese Journal of Organic Chemistry, 2006, 26, 27-42.

2005

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Efficient construction of novel alpha-keto spiro ketal and the total synthesis of (+/-)-terreinol
Wei Wan-Guo, Zhang Y.-X., Yao Zhu-Jun
Tetrahedron, 2005, 61, 11882-11886.


Preparation of enantiomerically pure 2-(1 '-aminomethyl)furan derivatives and synthesis of an unnatural polyhydroxylated piperidine
Cong X., Liu K.-G., Liao J., Yao Zhu-Jun
Tetrahedron Letters, 2005, 46, 8567-8571.


An iterative acetylene-epoxide coupling strategy for the total synthesis of longimicin C
He Y.-T., Xue S., Hu T.-S., Yao Zhu-Jun
Tetrahedron Letters, 2005, 46, 5393-5397.


Synthesis studies toward chloroazaphilone and vinylogous gamma-pyridones: Two common natural product core structures
Wei Wan-Guo, Yao Zhu-Jun
Journal of Organic Chemistry, 2005, 70, 4585-4590.


Chemoselective deprotection of cyclic N,O-aminals using catalytic bismuth(III) bromide in acetonitrile
Cong X., Hu F., Liu K.-G., Liao Q.-J., Yao Zhu-Jun
Journal of Organic Chemistry, 2005, 70, 4514-4516.


Macrocyclization studies and total synthesis of cyclomarin C, an anti-inflammatory marine cyclopeptide
Wen S.-J., Hu T.-S., Yao Zhu-Jun
Tetrahedron, 2005, 61, 4931-4938.


Stereoselective synthesis of new modified conformationally constrained L-tyrosine analogue with potential applications to SH2 domain ligands
Liu F., Hu T.-S., Yao Zhu-Jun
Tetrahedron, 2005, 61, 4971-4981.


Synthesis of a tetra-deuterium-labeled derivative of potent and selective anticancer agent AA005
Liu H.-X., Yao Zhu-Jun
Tetrahedron Letters, 2005, 46, 3525-3528.


Synthesis of two naturally occurring 4-hydroxylated butenolides with PTP1B inhibitory activity
Zhao Y., Jiang S., Guo Y.-W., Yao Zhu-Jun
Chinese Journal of Chemistry, 2005, 23, 173-175.

2004

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A chiron-based approach for the synthesis of tricyclic tyrosine analogue
Liu F., Jiao J., Zha H.-Y., Yao Zhu-Jun
Chinese Journal of Chemistry, 2004, 22, 1022-1028.

RCM approaches toward the diastereoselective synthesis of vicinal trans-diaminocyclitols from L-serine
Cong X., Liao Q.-J., Yao Zhu-Jun
Journal of Organic Chemistry, 2004, 69, 5314-5321.


Total synthesis of cyclomarin C
Wen S.-J., Yao Zhu-Jun
Organic Letters, 2004, 6, 2721-2724.


Synthesis of 4-azido-4-deoxy-Neu5,7,8,9Ac(4)2en1Me. A key intermediate for the synthesis of GG167 from D-glucono-delta-lactone
Liu K.-G., Yan S., Wu Y.-L., Yao Zhu-Jun
Organic Letters, 2004, 6, 2269-2272.


Synthesis of (2R,3aR,8aR)-6-chloro-3a-hydroxy-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indole-2-carboxylic acid methyl ester by reductive cyclization
Hong W.-X., Yao Zhu-Jun
Chinese Journal of Chemitry, 2004, 22, 365-370.

Parallel fragment assembly strategy towards multiple-ether mimicry of anticancer annonaceous acetogenins
Jiang S., Li Y., Chen X.-G., Hu T.-S., Wu Y.-L., Yao Zhu-Jun
Angewandte Chemie-International Edition, 2004, 43, 329-334.


2003

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Synthesis of a new stable conformationally constrained 2,7-anhydrosialic acid derivative
Liu K.-G., Zhou H.-B., Wu Y.-L., Yao Zhu-Jun
Journal of Organic Chemistry, 2003, 68, 9528-9531.


Studies on the synthesis of (2S,3R)-3-hydroxy-3-methylproline via C-2-N bond formation
Shen J.-W., Qin D.-G., Zhang H.-W., Yao Zhu-Jun
Journal of Organic Chemistry, 2003, 68, 7479-7484.


Synthesis of a new conformation-constrained L-tyrosine, analogue as a potential scaffold for SH2 domain ligands
Liu F., Zha H.-Y., Yao Zhu-Jun
Journal of Organic Chemistry, 2003, 68, 6679-6684.


A practical procedure for multisubstituted beta-naphthols and their derivatives
Wei W.-G., Yao Zhu-Jun
Tetrahedron, 2003, 59, 6621-6625.


An efficient enantioselective synthesis of the acyl side chain of polyoxypeptins
Qin D.-G., Yao Zhu-Jun
Tetrahedron Letters, 2003, 44, 571-574.


2002

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Synthesis of a mimicking hybrid of Annonaceous acetogenin with steroid for antitumoral activity investigation
Jiang S., Wu Y.-L., Yao Zhu-Jun
Chinese Journal of Chemistry, 2002, 20, 1393-1400.

Sharpless AD strategy toward the gamma-methyl butenolide unit of acetogenins: enantioselective synthesis of butenolide I and II with mosquito larvicidal activity
He Y.-T., Yang H.-N., Yao Zhu-Jun
Tetrahedron, 2002, 58, 8805-8810.


Recent progress of the synthetic study on sialic acid (N-acetylneuaminic acid) and its analogs
Li L.-S., Liu K.-G., Yao Zhu-Jun, Wu Yu-Lin
Chinese Journal of Organic Chemistry, 2002, 22, 718-734.

A new synthesis of Neu5Ac from D-glucono-delta-lactone
Liu Ke-Gang, Yan Shi, Wu Yu-Lin, Yao Zhu-Jun
Journal of Organic Chemitry, 2002, 67, 6758-6763.


Synthesis of a fully protected (2S,3R)-N-(1 ',1 '-dimethyl-2 '-propenyl)-3-hydroxytryptophan from tryptophan
Wen S.-J., Zhang H.-W., Yao Zhu-Jun
Tetrahedron Letters, 2002, 43, 5291-5294.


First synthesis of mosquito larvicidal butenolides I and II
Jiang S., Wu Yu-Lin, Yao Zhu-Jun
Chinese Journal of Chemistry, 2002, 20, 692-696.

Mimicry of annonaceous acetogenins: Enantioselective synthesis of a (4R)-hydroxy analogue having potent antitumor activity
Jiang Sheng, Liu Hai-Zhong, Sheng Gang, Zeng Bu-Bing, Cheng Xiao-Guang, Wu Yu-Lin, Yao Zhu-Jun
Journal of Organic Chemistry, 2002, 67, 3404-3408.


Enantioselective synthesis of (2S,3R)-3-hydroxy-3-methylproline, a novel amino acid found in polyoxypeptins
Qin Dong-Guang, Zha Hui-Yan, Yao Zhu-Jun
Journal of Organic Chemitry, 2002, 67, 1038-1040.


Electronic effect of indolecarboxaldehyde in the condensation with t-butyl bromoacetate promoted by biazaborolidine
Wen S.-J., Yao Zhu-Jun
Acta Chimica Sinica, 2002, 60, 129-133.

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List of Publications before 2002

  1.    Wu, P., Chen,W.-S., Hu, T.-S., Yao, Z.-J., Wu, Y.-L. Annonaceous Acetogenin from Annona Atemoya Seeds. J. Asian Nat. Prod. Research 2001, 3, 177.

  2.    Wu, Y.-L., Wu, W.-L., Yao, Z.-J., Li, Y.-L., Wang, Y.-F., Li, J.-C., Sun, X.-L., Peng, Z.-H., Yu, Q., Hu, T.-S., Zeng, B.-B., Wang, X.-Z. Syntheses of Enantiopure Natural Products from Sugars. Chinese J. Org. Chem. 2001, 21, 1051.

  3.    Atabey, N.; Gao, Y.; Yao, Z.-J.; Brechenridge, D.; Soon, L.; Burke Jr., T.R.; Bottaro, D.P. Potent blockade of hepatocyte growth factor-stimulated cell motility by selective inhibitors of Grb2-c-Met interaction. J. Biol. Chem. 2001, 276, 14308-14314.

  4.    Burke Jr., T. R., Yao, Z.-J., Ye, B., Miyoshi, K., Otaka, A., Wu., L., Zhang, Z.-Y. Phospho-azatyrosine, a less effective protein-tyrosine phosphatase substrate than phosphotyrosine. Bioorganic & Medicinal Chemistry Letters 2001, 11, 1265-8.

  5.    Burke Jr.,T. R., Yao, Z.-J., Gao, Y., Wu, J. X., Zhu, X., Luo, J. H., Guo, R., Yang, D. N-Terminal Carboxyl and Tetrazole-Containing Amides as Adjuvants to Grb2 SH2 Domain Ligand Binding. Bioorg. Med. Chem. 2001, 9, 1439-1445.

  6.    Burke Jr., T. R., Yao, Z.-J., Liu, D.-G., Voigt, J., Gao, Y. Phosphoryltyrosyl Mimetics in the Design of Peptide-Based Signal Transduction Inhibitors. Biopolymers 2001, 60, 32-44.

  7.    Zhang, Y.-L., Yao, Z.-J., Sarmiento, M., Wu, L., Burke, Jr., T. R., Zhang, Z.-Y. Isothermal Titration Calorimetric Study of Ligand Binding to Protein-Tyrosine Phosphatase 1B and Its Substrate-Trapping Mutants. J. Biol. Chem. 2000, 275(44), 34205-34212.

  8.    Long, Y.-Q., Lung, F.-D. T., Voigt, J. H., Yao, Z.-J., Burke, Jr., T. R., Yang, D., Luo, J. H., Guo, R., King, C. K., Roller, P. P. High affinity nonphosphorylated cyclic peptide inhibitors of Grb2-SH2 / growth factor receptor interactions. In Peptides: Frontier of Peptide Science, Proc. of 16th American Peptide Symposium, Tam, J. P., and Kaumaya, P. T. P. (Eds), ESCOM/Kluwer Acad. Publishers, Dordect, The Netherlands, 2000, 568-570.

  9.    Yao, Z.-J., Barchi, J. J., Burke, Jr., T. R. Design and synthesis of a new tyrosine analogue having c1 and c2 angles constrained to values observed for an SH2 domain-bound phosphotyrosyl residue. In Peptides for the New Millennium: Proc. of 16th American Peptide Symposium, Fields, G. B., Tam, J. P., and Barany, G. (Eds), Kluwer Acad. Publishers, Dordect, The Netherlands, 2000, p576-8.

  10.  Gao, Y., Yao, Z.-J., Voigt, J. H., Luo, J. H., Yang, D., Burke, Jr., T. R. Novel phosphotyrosyl mimetics for the preparation of potent small molecule Grb2 SH2 domain inhibitors. In Peptides for the New Millennium: Proc. of 16th American Peptide Symposium, Fields, G. B., Tam, J. P., and Barany, G. (Eds), Kluwer Acad. Publishers, Dordect, The Netherlands, 2000, p566-7.

  11.  Gao, Y., Luo, J., Yao, Z.-J., Guo, R., Zou, H., Kelley, J., Voigt, J. H., Yang, D., Burke, Jr.,  T. R.  Inhibition of Grb2 SH2 Domain Binding by Non-Phosphate Containing Ligands 2. 4-(2-Malonyl)phenylalanine as a potent Phosphotyrosyl Mimetic. J. Med. Chem. 2000, 43, 911-920.

  12.  Burke Jr., T.R.; Gao, Y.; Yao, Z.-J.; Voigt, J.; Luo, J.; Dajun, Y. Potent non phosphate- containing Grb2 SH2 domain inhibitors. Peptide Chemistry 1999. Proceedings of the 36th Japanese Peptide Symposium, Ed. by N. Fujii, The Japanese Peptide Society, 2000, pp 49-52.

  13.  Yao, Z.-J., Wu, H.-P., Wu, Y.-L. Polyether Mimics of Natural Occurring Cytotoxic Annonaceous Acetogenins. J. Med. Chem. 2000, 43, 2484-2487.

  14.  Liu, D.-G.; Yao, Z.-J.; Gao, Y.; Burke, T.R., Jr. Large scale preparation of cell permeable, non-phosphate containing Grb2 SH2 domain inhibitors. Organic Preparations and Procedures International 2000, 32, 197-201.

  15.  Chen, H., Cong, L.-N., Li, Y., Yao, Z.-J., Wu, L., Zhang, Z.-Y., Burke Jr., T. R., Quon, M. J. A Phosphotyrosyl Mimetic Peptide Reverses Impairment of Insulin-stimulated Translocation of Glut4 Caused by Overexpression of PTP1B in Rat Adipose Cells. Biochemistry 1999, 38(1), 384-389.

  16.  Yao, Z.-J., King, C. R., Cao, T., Kelley, J., Milne, G. W. A., Voigt, J. H., Burke Jr., T. R. Potent Inhibition of Grb2 SH2, Domain Binding by Non-Phosphate Cotaining Ligands. J. Med. Chem. 1999, 42(1), 25-35.

  17.  Burke Jr., T. R., Luo, J., Yao, Z.-J., Gao, Y., Milne, G. W. A., Voigt, J. H., King, C. R., Yang, D. Monocarboxylic-Based Phosphotyrosyl Mimetics in the Design of Grb2 SH2 Domain Inhibitors. Bioorganic and Medicinal Chemistry Lett. 1999, 9, 347-352.

  18.  Yao, Z.-J., Gao, Y., Voigt, J. H., Ford, Jr., H., Burke Jr., T. R. Synthesis of Fmoc-Protected 4-Carboxydifluoromethyl-L-phenylalanine: A Phosphotyrosyl Mimetic of Potential Use for Signal Transduction Studies. Tetrahedron. 1999, 55, 2865-2874.

  19.  Yu, Q., Yao, Z.-J., Chen, X.-G., Wu, Y.-L. Total Synthesis of (10R) and (10S)-corossolin, Determination of the C-10 configuration and the Unexpected Differential Toxicity toward Cancer Cell Caused by the Configuration at C-10. J. Org. Chem. 1999, 64, 2440-2445.

  20.  Long, Y.-Q., Yao, Z.-J., Lung, F.-D. T., Voigt, J. H., King, C. R., Burke, Jr., T. R., Roller, P. P. Overlapping function of amino acids in position-2 and Y0 leading to high affinity nonphosphorylated peptide ligands of Grb2-SH2 domain. Biochem. Biphys. Res. Comm. 1999, 264, 902-908.

  21.  Yao, Z.-J., Gao, Y., Burke, T. R., Jr. Preparation of L-N-Fmoc-Pmp(tBu2)-OH From L-Tyrosine. Tetrahedron: Asymmetry 1999, 10, 3727-3734.

  22.  Wu, Y.-L., Chen, H.-B., Jiang, K., Li, Y., Shan, F., Wang, D.-Y., Wang, Y.-F., Wu, W.-M., Wu, Y., Yao, Z.-J., Yue, Z.-Y., Zhou, C.-M. Interaction of biomolecules with qinghaosu (artemisinin) and its derivatives in the presence of ferrous ion C an exploration of antimalarial mechanism. Pure Appl. Chem. 1999, 71, 1139-1142.

  23.  Burke, T. R., Jr., Gao, Y., Yao, Z.-J., Voigt, J., Luo, J., Yang, D. Potent non phosphate-containing Grb2 SH2 domain inhibitors. Pept. Sci. 1999, 36, 49-52.

  24.  Wu, W.-M., Wu, Y., Wu, Y.-L., Yao, Z.-J., Zhou, C.-M., Li, Y., Shan, F. Unified Mechanism Framework for the Fe(II)-Induced Cleavage of Qinghaosu and Derivatives /Analogs. The First Spin-Trapping Evidence for the previously Postulated Secondary C-4 Radical. J. Am. Chem. Soc. 1998, 120, 3316-3325.

  25.  Hu, Y.-J., Huang, X.-D., Yao, Z.-J., Wu, Y.-L. Formal Synthesis of 3-Deoxy-D-manno-2-Octulosonic Acid (KDO) via a Highly Double-Stereoselective Hetero Diels-Alder Reaction Directed by a (Salen)Co(II) Catalyst and Chiral Diene. J. Org. Chem. 1998, 63, 2456-2461.

  26.  Yao, Z.-J., Ye, B., Miyoshi, K., Otaka, A., Burke Jr., T. R. Preparation of phospho-L-azatyrosine suitably protected for the solid phase synthesis of signal transduction-related peptides. A correction. Synlett. 1998, 428-430.

  27.  Burke Jr., T. R., Yao, Z.-J., Zhao, H. Enantioselective Synthesis of Nonphosphorous- Containing Phosphotyrosyl Mimetics and Their Use in Peptide Synthesis. Tetrahedron, 1998, 54, 9981-9994.

  28.  Yao, Z.-J., Ye, B., Wu, X.-W, Wang, S., Wu, L., Zhang, Z.-Y., Burke Jr., T. R. Structure-based design and synthesis of small molecule protein-tyrosine phosphatase 1B inhibitors. Bioorganic and Medicinal Chemistry, 1998, 4, 1799-1810.

  29.  Tan, H.-T., Chen, W.-S., Yu, Q., Yao, Z.-J., Wu, Y.-L. The Isolation and Structure of Microcarpacin B. Youji Huaxue (Chin. J. Org. Chem.) 1998, 18(3), 219.

  30.  Groves, M. R., Yao, Z.-J., Roller, P. P., Burke Jr., T. R., Barford, D. Structral Basis for Inhibition of the Protein Tyrosine Phosphatase 1B by Phosphotyrosine Peptide Mimetics. Biochemstry 1998, 37(51), 17773-17783.

  31.  Chen, W.-S., Yao, Z.-J., Wu, Y.-L. Annonaceous acetogenins from Uvaria microcarpa Seeds. The isolation and structure of microcarpacin. Acta Chemica Sinica 1997, 55, 723-728.

  32.  Burke Jr., T. R., Yao, Z.-J., Smyth, M. S., Ye, B. Phosphotyrosyl-based motifs in the structure-based design of protein-tyrosine kinase-dependent signal transduction inhibitors. Current Pharmaceutical Design, 1997, 3, 291.

  33.  Ye, B., Yao, Z.-J., Burke Jr., T. R.  Synthesis of a new tyrosine analog having X1 and X2 angles constrained to values observed for SH2 domain-bound phosphotyrosyl residue. J. Org. Chem. 1997, 62, 5428.

  34.  Yao, Z.-J., Ye, B., Zhao, H., Yan, X., Wu, L., Barford, D., Wang, S., Zhang, Z.-Y., Burke Jr., T. R. Structure-based design of small molecule protein-tyrosine phosphatase inhibitors. In Peptides: Frontier of Peptide Science, Proc. of 15Th American Peptide Symposium, Tam, J. P., and Kaumaya, P. T. P. (Eds), ESCOM/Kluwer Acad. Publishers, Dordect, The Netherlands, 1997, pp183-185.

  35.  Chen, W.-S., Yao, Z.-J., Xu, Y.-Z., Zhang, Y.-B., Wu, Y.-L. Study on the annonaceous acetogenins from Annona Atemoya Hort. Youji Huaxue (Chin. J. Org. Chem.) 1996, 16, 145.

  36.  Yao, Z.-J., Yu, Q., Wu, Y.-L. Two-directional enantioselective synthesis of (+)-ancepsenolide. Synthetic Communication. 1996, 26, 3613.

  37.  Wu, W.-M., Yao, Z.-J., Wu, Y.-L., Jiang, K., Wang, Y.-F., Chen, H.-B., Shan, F., Li, Y. Ferrous ion induced cleavage of the peroxy bond in qinghaosu and its derivatives and the DNA damage associated with this process. Chemical Communication 1996, 2213.

  38.  Yao, Z.-J., Wu, Y.-L. Synthetic studies toward mono-THF annonaceous acetogenins, an enantioselective and convergent approach to corossolone and (10RS)-corossoline. J. Org. Chem. 1995, 60, 1170.

  39.  Wu, W.-L., Yao, Z.-J., Li, Y.-L., Li, J.-C., Xia, Y., Wu, Y.-L. Diastereoselective propargylation of -alkoxy aldehyde with propargyl bromide and zinc, a versatile and efficient method for synthesis of chiral oxygenated acyclic natural products. J. Org. Chem. 1995, 60, 3257.

  40.  Chen, W.-S., Yao, Z.-J., Zhang, Y.-B., Xu, Y.-Z., Wu, Y.-L. Atemoyacin A: a new bis-tetrahydrofuranyl annonaceous acetogenin from Annona Atemoya H. Chinese J. Chem. 1995, 13, 263.

  41.  Chen, W.-S., Yao, Z.-J., Wu, Y.-L. Study on the chemical constituents of Annona glabra Linn. Youji Huaxue (Chin. J. Org. Chem.) 1995, 15, 85.

  42.  Yao, Z.-J., Wu, Y.-L. Annonaceous acetogenins: Future stars against cancer. Youji Huaxue (Chin. J. Org. Chem.) 1995, 15, 120.

  43.  Chen, W.-S., Yao, Z.-J., Zhang, Y.-B., Xu, Y.-Z., Wu, Y.-L. Study on the chemical constituents of Annona Atemoya H. and the isolation and the structure of atemoyacin B. Acta Chemica Sinica 1995, 53, 516.

  44.  Li, J.-C., Li, Y.-L., Peng, Z.-H., Sun, X.-L., Wang, Y.-F., Wu, Y.-L., Yao, Z.-J. Chiral syntheses of acyclic natural products from sugars. J. Chin. Chem. Soc. (Taipei) 1995, 42, 681.

  45.  Yao, Z.-J., Wu, Y.-L. Total synthesis of (10RS, 15R, 16S, 20S, 34R)-corossoline. Tetrahedron Lett. 1994, 35, 157.

  46.   Yao, Z.-J., Zhang, Y.-B., Wu, Y.-L. Synthesis of annonaceous acetogenin (4S, 5S) and (4S, 5R)-muricatacin as well as confirmation of absolute configuration of the tetrahydrofuran segment of annonacin. Acta Chim. Sinica 1992, 50, 901.

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